SCHEMBL66535

SCHEMBL66535

O=C(C[C@@H](CO)N(Cc1ccccc1)C(=O)O)N(Cc1cccc(Cl)c1Cl)C1CC1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 7/20 0.52
SLC6A2 P23975 6/20 0.52
SLC6A3 Q01959 2/20 0.46
KCNH2 Q12809 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
REN P00797 8/20 0.44
GHSR Q92847 1/20 0.39
UBE2M P61081 1/20 0.39
DCUN1D1 Q96GG9 1/20 0.39
OPRM1 P35372 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
TACR1 P25103 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65406 0.81 REN (0.49) SLC6A4SLC6A2SLC6A3KCNH2CYP3A4
SCHEMBL65337 0.79 SLC6A4 (0.58) SLC6A4SLC6A2SLC6A3KCNH2CYP3A4
SCHEMBL79378 0.79 SLC6A4 (0.64) SLC6A4SLC6A2SLC6A3KCNH2CYP3A4
SCHEMBL65338 0.79 SLC6A4 (0.58) SLC6A4SLC6A2SLC6A3KCNH2CYP3A4
SCHEMBL79894 0.77 SLC6A4 (0.47) SLC6A4SLC6A2SLC6A3KCNH2CYP3A4
SCHEMBL65438 0.75 SLC6A4 (0.51) SLC6A4SLC6A2SLC6A3KCNH2CYP3A4
SCHEMBL5072329 0.74 SLC6A4 (0.59) SLC6A4SLC6A2SLC6A3KCNH2CYP3A4
SCHEMBL5072308 0.71 SLC6A4 (0.76) SLC6A4SLC6A2SLC6A3KCNH2CYP3A4
SCHEMBL8171105 0.71 SLC6A4 (0.59) SLC6A4SLC6A2SLC6A3KCNH2CYP3A4
SCHEMBL662533 0.71 SLC6A4 (0.53) SLC6A4SLC6A2SLC6A3KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed