SCHEMBL6655717

SCHEMBL6655717

CC#CCOc1ccc(SC(C(=O)O)c2cccc3ccccc23)cc1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 12/20 0.59
MMP9 P14780 4/20 0.44
MMP13 P45452 4/20 0.44
ALOX5 P09917 8/20 0.41
PTGES O14684 3/20 0.41
MMP1 P03956 2/20 0.41
PPARG P37231 6/20 0.40
PPARA Q07869 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6654293 0.89 ADAM17 (0.70) ADAM17MMP9MMP13MMP1
SCHEMBL6787275 0.85 ADAM17 (0.62) ADAM17MMP9MMP13ALOX5PTGES
SCHEMBL6657581 0.83 ADAM17 (0.78) ADAM17MMP9MMP13ALOX5MMP1
SCHEMBL6656809 0.81 ADAM17 (0.63) ADAM17MMP9MMP13ALOX5PTGES
SCHEMBL6657088 0.78 ADAM17 (0.65) ADAM17MMP9MMP13MMP1PPARA
SCHEMBL6656399 0.76 ADAM17 (0.62) ADAM17MMP9MMP13ALOX5PTGES
SCHEMBL6654467 0.76 ADAM17 (0.65) ADAM17MMP9MMP13ALOX5PTGES
SCHEMBL6659002 0.76 ADAM17 (0.77) ADAM17MMP9MMP13MMP1
SCHEMBL6661896 0.76 ALOX5 (0.46) ALOX5PTGESPPARG
SCHEMBL6658123 0.75 ADAM17 (0.64) ADAM17MMP9MMP13MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147080-B1 ALKYNYL CONTAINING HYDROXAMIC ACID COMPOUNDS AS TACE INHIBITORS WYETH CORP (US) 2004-07-21 EP disclosed