SCHEMBL6656239

SCHEMBL6656239

CCc1nc2c(OC)c(OC)ccc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 1/20 0.45
PDE3B Q13370 2/20 0.43
PDE3A Q14432 2/20 0.43
DDAH1 O94760 1/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAPT P10636 1/20 0.41
CYP1A2 P05177 2/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6654447 0.85 CACNA1H (0.42) CACNA1HPDE3BPDE3AKDM4EALDH1A1
SCHEMBL2431585 0.83 TSHR (0.47) PDE3BPDE3ADDAH1KDM4EALDH1A1
SCHEMBL6654775 0.78 PDE3B (0.43) CACNA1HPDE3BPDE3AKDM4EALDH1A1
SCHEMBL2269491 0.75 ADORA1 (0.50) PDE3BPDE3ADDAH1KDM4EMEN1
SCHEMBL6656241 0.74 PDE3B (0.50) PDE3BPDE3ADDAH1KDM4EALDH1A1
SCHEMBL6653651 0.72 TNKS (0.51) KDM4EALDH1A1MAPTHPGDHSD17B10
SCHEMBL22533865 0.71 DDAH1 (0.41) PDE3BPDE3ADDAH1ADORA3ADORA2A
SCHEMBL29424800 0.71 DDAH1 (0.41) PDE3BPDE3ADDAH1ADORA3ADORA2A
SCHEMBL9847093 0.69 CBFB (0.46) DDAH1TP53ADORA3ADORA2AADORA1
SCHEMBL6657269 0.68 DDAH1 (0.44) DDAH1ADORA3ADORA2AADORA1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1428510-A1 Dyeing composition comprising a tertiary paraphenylenediamine containing a pyrrolidine, and a heterocyclic coupler or a hydroxybenzamide ; method and use L'OREAL (FR) 2004-06-16 EP claimed
EP-1428510-A1 Dyeing composition comprising a tertiary paraphenylenediamine containing a pyrrolidine, and a heterocyclic coupler or a hydroxybenzamide ; method and use L'OREAL (FR) 2004-06-16 EP disclosed