SCHEMBL6656679

SCHEMBL6656679

CCNC(=O)c1ccc(C)c(-c2ccc(C(N)=O)cc2)c1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 20/20 0.67
HSPB1 P04792 1/20 0.51
CYP2C9 P11712 1/20 0.51
MAPK11 Q15759 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5488332 0.87 MAPK14 (0.59) MAPK14HSPB1CYP2C9MAPK11
SCHEMBL6275051 0.85 MAPK14 (0.54) MAPK14HSPB1CYP2C9MAPK11
SCHEMBL3374385 0.79 EPHX2 (0.56)
SCHEMBL13702344 0.78 AOC3 (0.54)
SCHEMBL6655486 0.78 S1PR4 (0.67) MAPK14
SCHEMBL13146376 0.78 MAPK14 (0.79) MAPK14HSPB1CYP2C9MAPK11
SCHEMBL5633482 0.76 MAPK14 (0.77) MAPK14HSPB1CYP2C9MAPK11
SCHEMBL6658772 0.76 MAPK14 (0.74) MAPK14CYP2C9MAPK11
SCHEMBL6748200 0.76 MAPK14 (0.77) MAPK14HSPB1CYP2C9MAPK11
SCHEMBL4151138 0.76 NR1H4 (0.61) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1435933-A1 5'-CARBAMOYL-2'-METHYL-1,1'-BIPHENYL-4-CARBOXAMIDE DERIVATIVES AND THEIR USE AS P38 KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2004-07-14 EP disclosed
WO-2003032970-A1 5'-CARBAMOYL-2'-METHYL-1,1'-BIPHENYL-4-CARBOXAMIDE DERIVATIVES AND THEIR USE AS P38 KINASE INHIBITORS GLAXO GROUP LIMITED (GB) 2003-04-24 WO disclosed