SCHEMBL6660879

SCHEMBL6660879

Fc1ccc(/C=C/c2ncnc3[nH]cnc23)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 1/20 0.46
IP6K3 Q96PC2 1/20 0.46
NFE2L2 Q16236 6/20 0.38
GRM4 Q14833 1/20 0.38
PDPK1 O15530 1/20 0.38
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 2/20 0.37
KMT2A Q03164 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
MAPKAPK2 P49137 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
MKNK1 Q9BUB5 1/20 0.35
APP P05067 1/20 0.34
PTGS1 P23219 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6660882 1.00 IP6K1 (0.46) IP6K1IP6K3NFE2L2GRM4PDPK1
SCHEMBL6663881 0.84 MEN1 (0.47) IP6K1IP6K3GRM4PDPK1KDM4E
SCHEMBL6663884 0.84 MEN1 (0.47) IP6K1IP6K3GRM4PDPK1KDM4E
SCHEMBL4065715 0.76 TRPA1 (0.51) IP6K1IP6K3NFE2L2GRM4KDM4E
SCHEMBL4065710 0.76 TRPA1 (0.51) IP6K1IP6K3NFE2L2GRM4KDM4E
SCHEMBL31060480 0.76 MKNK1 (0.51) IP6K1IP6K3PDPK1KDM4EMEN1
SCHEMBL3468490 0.71 GSK3A (0.53) KDM4EMAPTKMT2AL3MBTL1GAA
SCHEMBL3468495 0.71 GSK3A (0.53) KDM4EMAPTKMT2AL3MBTL1GAA
SCHEMBL6662321 0.71 ADORA1 (0.44) IP6K1IP6K3NFE2L2KDM4EMEN1
SCHEMBL6662325 0.71 ADORA1 (0.44) IP6K1IP6K3NFE2L2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444982-A1 The use of purine derivatives as selective kinase inhibitors MERCKLE GMBH (DE) 2004-08-11 EP disclosed