SCHEMBL6661082

SCHEMBL6661082

COC(=O)/C=C(/N)c1ccc(OC)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.66
MAPK1 P28482 1/20 0.66
HSD17B10 Q99714 1/20 0.66
CA1 P00915 6/20 0.58
CA2 P00918 6/20 0.58
PARP10 Q53GL7 2/20 0.58
PARP1 P09874 1/20 0.58
PARP2 Q9UGN5 1/20 0.58
PARP4 Q9UKK3 1/20 0.58
PDE4A P27815 1/20 0.54
PDE4B Q07343 1/20 0.54
PDE4C Q08493 1/20 0.54
PDE4D Q08499 1/20 0.54
CES2 O00748 1/20 0.52
CES1 P23141 1/20 0.52
PLK1 P53350 1/20 0.50
PRSS1 P07477 1/20 0.48
PRSS2 P07478 1/20 0.48
PRSS3 P35030 1/20 0.48
NPC1 O15118 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7933746 1.00 RAB9A (0.66) RAB9AMAPK1HSD17B10CA1CA2
SCHEMBL6661088 1.00 RAB9A (0.66) RAB9AMAPK1HSD17B10CA1CA2
SCHEMBL6657569 0.84 TDP1 (0.52) RAB9AMAPK1HSD17B10PDE4APDE4B
SCHEMBL6657574 0.84 TDP1 (0.52) RAB9AMAPK1HSD17B10PDE4APDE4B
SCHEMBL30189391 0.83 MAPK1 (0.59) RAB9AMAPK1HSD17B10CA1CA2
SCHEMBL28810859 0.83 MAPK1 (0.59) RAB9AMAPK1HSD17B10CA1CA2
SCHEMBL2649166 0.82 SMN1; SMN2 (0.59) RAB9AMAPK1HSD17B10CA1CA2
SCHEMBL14691237 0.82 SMN1; SMN2 (0.59) RAB9AMAPK1HSD17B10CA1CA2
SCHEMBL7931260 0.82 RAB9A (0.45) RAB9AMAPK1HSD17B10PDE4APDE4B
SCHEMBL7931264 0.82 RAB9A (0.45) RAB9AMAPK1HSD17B10PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004011414-A1 E-ISOMERIC β-AROMATIC OR HETEROAROMATIC SUBSTITUTED β-ACYLAMINO-ACRYLATES AND METHODS OF PREPARING THE SAME DSM IP ASSETS B.V. (NL) 2004-02-05 WO disclosed