SCHEMBL6657569

SCHEMBL6657569

COC(=O)/C=C(/N)c1ccc(C)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.52
ALDH1A1 P00352 7/20 0.49
MAPT P10636 4/20 0.49
KDM4E B2RXH2 1/20 0.49
RAB9A P51151 5/20 0.46
MAPK1 P28482 1/20 0.46
HSD17B10 Q99714 1/20 0.46
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
PKM P14618 2/20 0.44
HTT P42858 2/20 0.44
ATM Q13315 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
LMNA P02545 2/20 0.44
HPGD P15428 2/20 0.44
GAA P10253 2/20 0.44
NLRP1 Q9C000 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6657574 1.00 TDP1 (0.52) TDP1ALDH1A1MAPTKDM4ERAB9A
SCHEMBL7933746 0.84 RAB9A (0.66) ALDH1A1RAB9AMAPK1HSD17B10PDE4A
SCHEMBL6661088 0.84 RAB9A (0.66) ALDH1A1RAB9AMAPK1HSD17B10PDE4A
SCHEMBL1928738 0.84 SMN1; SMN2 (0.59) ALDH1A1MAPTKDM4ERAB9AMAPK1
SCHEMBL14691237 0.84 SMN1; SMN2 (0.59) ALDH1A1MAPTKDM4ERAB9AMAPK1
SCHEMBL7931260 0.84 RAB9A (0.45) ALDH1A1MAPTKDM4ERAB9AMAPK1
SCHEMBL7931264 0.84 RAB9A (0.45) ALDH1A1MAPTKDM4ERAB9AMAPK1
SCHEMBL6661082 0.84 RAB9A (0.66) ALDH1A1RAB9AMAPK1HSD17B10PDE4A
SCHEMBL2649166 0.84 SMN1; SMN2 (0.59) ALDH1A1MAPTKDM4ERAB9AMAPK1
SCHEMBL7921709 0.83 TSHR (0.50) TDP1ALDH1A1MAPTKDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004011414-A1 E-ISOMERIC β-AROMATIC OR HETEROAROMATIC SUBSTITUTED β-ACYLAMINO-ACRYLATES AND METHODS OF PREPARING THE SAME DSM IP ASSETS B.V. (NL) 2004-02-05 WO disclosed