SCHEMBL6661151

SCHEMBL6661151

COC(=O)/C=C(/N)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.60
ALDH1A1 P00352 4/20 0.56
CES2 O00748 1/20 0.55
CES1 P23141 1/20 0.55
TP53 P04637 1/20 0.54
PRSS1 P07477 1/20 0.54
PRSS2 P07478 1/20 0.54
PRSS3 P35030 1/20 0.54
MAPT P10636 6/20 0.53
KMT2A Q03164 5/20 0.53
MEN1 O00255 4/20 0.53
POLB P06746 1/20 0.53
CTDSP1 Q9GZU7 1/20 0.53
HSP90AA1 P07900 1/20 0.53
HPGD P15428 1/20 0.53
MAPK1 P28482 1/20 0.53
CACNA1B Q00975 1/20 0.53
APBA1 Q02410 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
NLRP1 Q9C000 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6661153 1.00 TSHR (0.60) TSHRALDH1A1CES2CES1TP53
SCHEMBL16979582 0.86 ALDH1A1 (0.60) TSHRALDH1A1CES2CES1TP53
SCHEMBL16971093 0.86 ALDH1A1 (0.60) TSHRALDH1A1CES2CES1TP53
SCHEMBL7319345 0.83 ALDH1A1 (0.57) TSHRALDH1A1CES2CES1TP53
SCHEMBL14416438 0.82 ALDH1A1 (0.52) TSHRALDH1A1CES2CES1TP53
SCHEMBL563406 0.81 TP53 (0.52) TSHRALDH1A1CES2CES1TP53
SCHEMBL21457629 0.81 ALDH1A1 (0.51) TSHRALDH1A1CES2CES1TP53
SCHEMBL10539195 0.81 ALDH1A1 (0.58) TSHRALDH1A1CES2CES1TP53
SCHEMBL27575567 0.79 TSHR (0.64) TSHRALDH1A1CES2CES1TP53
SCHEMBL14188168 0.79 PARP1 (0.56) KMT2AMEN1POLBRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004011414-A1 E-ISOMERIC β-AROMATIC OR HETEROAROMATIC SUBSTITUTED β-ACYLAMINO-ACRYLATES AND METHODS OF PREPARING THE SAME DSM IP ASSETS B.V. (NL) 2004-02-05 WO disclosed
US-4990507-A Cardiotonic agents FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-02-05 US disclosed
EP-0228845-B1 N-CONTAINING HETEROCYCLIC COMPOUNDS, PROCESSES FOR THE PREPARATION THEREOF AND COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1990-12-12 EP disclosed
US-4931453-A CARDIOVASCULAR, HYPOTENSIVE AGENTS FUJISAWA PHARMACEUTICAL COMPANY, LTD. (JP) 1990-06-05 US disclosed
US-4857527-A HYPOTENSIVE, ANTISCHEMIC AGENT FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-08-15 US disclosed
US-4831030-A FOR CEREBROVASCULAR DISEASES; HYPERTENSIVE AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1989-05-16 US disclosed
EP-0228845-A2 N-containing heterocyclic compounds, processes for the preparation thereof and composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1987-07-15 EP disclosed