SCHEMBL7319345

SCHEMBL7319345

COC(=O)C=C(C(C)=O)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.57
CES2 O00748 1/20 0.53
CES1 P23141 1/20 0.53
TP53 P04637 1/20 0.51
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
MAPT P10636 4/20 0.51
HSP90AA1 P07900 1/20 0.51
HPGD P15428 1/20 0.51
MAPK1 P28482 1/20 0.51
CACNA1B Q00975 1/20 0.51
APBA1 Q02410 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
NLRP1 Q9C000 1/20 0.51
RAB9A P51151 4/20 0.50
TSHR P16473 2/20 0.50
NPC1 O15118 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.48
SETD7 Q8WTS6 1/20 0.48
HTT P42858 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16971093 0.86 ALDH1A1 (0.60) ALDH1A1CES2CES1TP53MEN1
SCHEMBL16979582 0.86 ALDH1A1 (0.60) ALDH1A1CES2CES1TP53MEN1
SCHEMBL7312492 0.86 GLO1 (0.54) ALDH1A1CES2CES1TP53MEN1
SCHEMBL6661151 0.83 TSHR (0.60) ALDH1A1CES2CES1TP53MEN1
SCHEMBL6661153 0.83 TSHR (0.60) ALDH1A1CES2CES1TP53MEN1
SCHEMBL7275168 0.82 ALDH1A1 (0.49) ALDH1A1CES2CES1TP53MEN1
SCHEMBL14416438 0.80 ALDH1A1 (0.52) ALDH1A1CES2CES1TP53MEN1
SCHEMBL563406 0.79 TP53 (0.52) ALDH1A1CES2CES1TP53MEN1
SCHEMBL21457629 0.79 ALDH1A1 (0.51) ALDH1A1CES2CES1TP53MEN1
SCHEMBL10539195 0.79 ALDH1A1 (0.58) ALDH1A1CES2CES1TP53MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0183848-B1 POLYAZAHETEROCYCLIC DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITION Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1990-09-12 EP disclosed
US-4918074-A CALCIUM ANTAGONISTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1990-04-17 US disclosed
EP-0217142-A2 A polyazaheterocyclic compound Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1987-04-08 EP disclosed
EP-0183848-A1 POLYAZAHETEROCYCLIC DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITION Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1986-06-11 EP disclosed