SCHEMBL6662818

SCHEMBL6662818

OB(O)Oc1ccc(COCc2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.58
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
PTGS1 P23219 1/20 0.46
SLC6A2 P23975 1/20 0.46
CYP2C19 P33261 1/20 0.46
PTGS2 P35354 1/20 0.46
SLC6A3 Q01959 1/20 0.46
HIF1A Q16665 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
LTA4H P09960 1/20 0.42
EPHX2 P34913 1/20 0.42
MAOB P27338 2/20 0.42
BCHE P06276 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
FFAR1 O14842 1/20 0.41
FFAR4 Q5NUL3 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6660289 0.88 TDP1 (0.50) TSHRLMNACYP1A2PTGS1SLC6A2
SCHEMBL4768663 0.88 TDP1 (0.50) TSHRLMNACYP1A2PTGS1SLC6A2
SCHEMBL1373373 0.85 LMNA (0.66) LMNACYP1A2PTGS1SLC6A2CYP2C19
SCHEMBL5370037 0.84 TSHR (0.48) TSHRLMNACYP1A2PTGS1SLC6A2
SCHEMBL16320997 0.84 LMNA (0.47) TSHRLMNACYP1A2PTGS1SLC6A2
SCHEMBL28077460 0.84 LTA4H (0.55) LMNACYP1A2CYP2C19LTA4HL3MBTL1
SCHEMBL6661512 0.83 IDO1 (0.50) HDAC6MAOBL3MBTL1TDP1CA1
SCHEMBL27781804 0.83 LMNA (0.58) LMNACYP1A2PTGS1SLC6A2CYP2C19
SCHEMBL5373560 0.82 TSHR (0.50) TSHRLMNACYP1A2PTGS1SLC6A2
SCHEMBL5377522 0.81 TSHR (0.48) TSHRLMNACYP1A2PTGS1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104230971-B Boric acid and ester as inhibitors of fatty amide hydrolase 英菲尼提制药公司 2017-11-24 CN disclosed
CN-101863913-B Preparation method of fluorinated aryl-containing boron compound SHANGHAI RES INST CHEMICAL IND 2013-02-27 CN disclosed
CN-101863913-A Preparation method of fluorinated aryl-containing boron compound SHANGHAI RES INST CHEMICAL IND 2010-10-20 CN disclosed
CN-101563089-A Boronic acids and esters as inhibitors of fatty amide hydrolase INFINITY DISCOVERY INC (US) 2009-10-21 CN disclosed
EP-1444981-A1 INTRACELLULAR CALCIUM CONCENTRATION INCREASE INHIBITORS Mikoshiba, Katsuhiko (JP) 2004-08-11 EP disclosed
EP-0743943-B1 PYRIDYL IMIDAZOLE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF KOREA RES INST CHEM TECH (KR) 2001-10-31 EP disclosed
US-5849753-A Pyridyl imidazole derivatives and processes for the preparation thereof KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1998-12-15 US disclosed
EP-0743943-A1 PYRIDYL IMIDAZOLE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1996-11-27 EP disclosed
WO-1995021838-A1 PYRIDYL IMIDAZOLE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1995-08-17 WO disclosed