SCHEMBL6663355

SCHEMBL6663355

Oc1ccc2nc(-c3ccc(F)cc3)c(-c3ccccc3)cc2c1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
PSMB5 P28074 1/20 0.52
DHODH Q02127 7/20 0.48
ESR1 P03372 3/20 0.47
ESR2 Q92731 3/20 0.47
ADORA1 P30542 2/20 0.47
ADORA2A P29274 1/20 0.44
EGFR P00533 1/20 0.44
MAPK14 Q16539 1/20 0.44
PDE10A Q9Y233 1/20 0.44
APP P05067 1/20 0.43
SULT1A1 P50225 1/20 0.43
AKT1 P31749 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8956599 0.83 PSMB5 (0.52) PSMB5DHODHADORA1MAPK14AKT1
SCHEMBL9692642 0.79 KMT2A (0.69) MEN1KMT2ADHODHESR2MAPK14
SCHEMBL7155536 0.79 KMT2A (0.69) MEN1KMT2ADHODHESR2MAPK14
SCHEMBL6662378 0.77 DHODH (0.50) MEN1KMT2ADHODHESR1ESR2
SCHEMBL6662078 0.75 ESR1 (0.73) MEN1KMT2ADHODHESR1ESR2
SCHEMBL28037634 0.75 KMT2A (0.79) MEN1KMT2AESR1ESR2
SCHEMBL28037189 0.75 KMT2A (0.79) MEN1KMT2AESR1ESR2
SCHEMBL6665512 0.74 ADORA1 (0.47) MEN1KMT2ADHODHADORA1ADORA2A
SCHEMBL3626800 0.74 PSMB5 (0.45) MEN1KMT2APSMB5DHODHESR1
SCHEMBL8956354 0.74 KDM4E (0.51) PSMB5DHODHADORA1MAPK14PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861864-B1 Method of preparation of polyquinolines HITACHI CHEMICAL CO LTD (JP) 2004-08-25 EP disclosed
EP-0861864-A2 Method of preparation of polyquinolines HITACHI CHEMICAL CO., LTD. (JP) 1998-09-02 EP disclosed
US-5786071-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-07-28 US disclosed
US-5723573-A ACETYLENIC END GROUPS HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-03-03 US disclosed
US-5648448-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1997-07-15 US disclosed