SCHEMBL6665512

SCHEMBL6665512

Oc1cccc2cc(-c3ccccc3)c(-c3ccc(F)cc3)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.47
KDM4E B2RXH2 3/20 0.47
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
TOP1 P11387 2/20 0.41
GRM2 Q14416 2/20 0.40
TNKS O95271 1/20 0.40
PARP1 P09874 1/20 0.40
TNKS2 Q9H2K2 1/20 0.40
ALOX5 P09917 1/20 0.40
GPR84 Q9NQS5 1/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
PDE10A Q9Y233 1/20 0.39
NPC1 O15118 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
DHODH Q02127 1/20 0.39
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10913571 0.91 KDM4E (0.54) ADORA1KDM4EHSD17B1HSD17B2ADORA3
SCHEMBL6256195 0.78 KDM4E (0.57) KDM4ETNKSPARP1TNKS2KMT2A
SCHEMBL2274802 0.76 KDM4E (0.49) ADORA1KDM4EHSD17B1HSD17B2ADORA3
SCHEMBL6663355 0.74 MEN1 (0.53) ADORA1ADORA2AKMT2AMEN1PDE10A
SCHEMBL7120189 0.74 PDE10A (0.57) ADORA1KDM4EADORA2AKMT2AMEN1
SCHEMBL7755155 0.74 KDM4E (0.49) ADORA1KDM4EHSD17B1HSD17B2ADORA3
SCHEMBL28304915 0.72 PSMB5 (0.42) ADORA1KDM4EADORA3ADORA2APDE10A
SCHEMBL29963685 0.71 MAPK14 (0.45) ADORA1KDM4EADORA2ATOP1GRM2
SCHEMBL27703790 0.71 KDM4E (0.47) ADORA1KDM4EADORA3ADORA2AKMT2A
SCHEMBL2858652 0.71 KDM4E (0.49) KDM4EKMT2AMEN1PDE10ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861864-B1 Method of preparation of polyquinolines HITACHI CHEMICAL CO LTD (JP) 2004-08-25 EP disclosed
EP-0861864-A2 Method of preparation of polyquinolines HITACHI CHEMICAL CO., LTD. (JP) 1998-09-02 EP disclosed
US-5786071-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-07-28 US disclosed
US-5723573-A ACETYLENIC END GROUPS HITACHI CHEMICAL COMPANY, LTD. (JP) 1998-03-03 US disclosed
US-5648448-A Method of preparation of polyquinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1997-07-15 US disclosed