SCHEMBL6665941

SCHEMBL6665941

NS(=O)(=O)c1ccc(-n2ncc3c2-c2ccsc2CC3)cc1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 11/20 0.61
CA9 Q16790 11/20 0.61
CA4 P22748 10/20 0.61
CA1 P00915 10/20 0.61
CA12 O43570 6/20 0.54
CA3 P07451 5/20 0.54
CA6 P23280 5/20 0.54
CA5A P35218 5/20 0.54
CA7 P43166 5/20 0.54
CA13 Q8N1Q1 5/20 0.54
CA14 Q9ULX7 5/20 0.54
CA5B Q9Y2D0 5/20 0.54
IKBKB O14920 1/20 0.49
PTGS2 P35354 8/20 0.46
PTGS1 P23219 6/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13238794 0.76 PTGS2 (0.47) CA2CA9CA4CA1CA12
SCHEMBL6659189 0.74 CCNA2 (0.64) CA2CA9CA4CA1IKBKB
SCHEMBL14747600 0.74 PTGS2 (0.69) PTGS2PTGS1
SCHEMBL3107038 0.70 CA2 (0.65) CA2CA9CA4CA1CA12
SCHEMBL6660718 0.69 CA9 (0.55) CA2CA9CA4CA1CA12
SCHEMBL6632506 0.68 CA2 (0.50) CA2CA9CA4CA1CA12
Hydrochloric Acid SCHEMBL7939254 0.65 PLK4 (0.39) IKBKB
SCHEMBL8765473 0.64 PTGS2 (0.76) CA2CA9CA4CA1CA12
SCHEMBL8764591 0.64 PTGS2 (0.64) CA2CA9CA4CA1CA12
SCHEMBL8765113 0.64 PTGS2 (0.62) CA2CA9CA4CA1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1476431-A1 TRICYCLIC PYRAZOLE DERIVATIVES FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2004-11-17 EP claimed
WO-2003070706-A1 TRICYCLIC PYRAZOLE DERIVATIVES FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2003-08-28 WO claimed