SCHEMBL6667068

SCHEMBL6667068

Cc1ccc(-c2ccccc2)c(C(=O)Nc2ccc3c(c2)CCN3C(=O)Cc2cscn2)c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.43
TP53 P04637 2/20 0.43
RAB9A P51151 2/20 0.43
NPC1 O15118 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CREBBP Q92793 1/20 0.40
POLB P06746 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
AVPR2 P30518 4/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
EIF2AK3 Q9NZJ5 2/20 0.38
EIF2AK1 Q9BQI3 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
AVPR1A P37288 2/20 0.38
PDE7A Q13946 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6804945 0.91 MAPT (0.46) MAPTTP53RAB9ANPC1SMN1; SMN2
SCHEMBL6663855 0.88 SRPK1 (0.43) MAPTTP53LMNAHTR2AHTR2C
SCHEMBL6664878 0.88 EIF2AK3 (0.48) MAPTTP53RAB9ANPC1SMN1; SMN2
SCHEMBL6670249 0.86 MAPT (0.42) MAPTTP53RAB9ANPC1SMN1; SMN2
SCHEMBL6669291 0.85 MAPT (0.48) MAPTTP53RAB9ANPC1SMN1; SMN2
SCHEMBL6667964 0.85 EIF2AK3 (0.50) MAPTTP53RAB9ANPC1SMN1; SMN2
SCHEMBL6671845 0.84 CYP11B1 (0.43) MAPTTP53RAB9ANPC1SMN1; SMN2
SCHEMBL6665119 0.84 EIF2AK3 (0.44) MAPTTP53RAB9ANPC1SMN1; SMN2
SCHEMBL6803919 0.83 EIF2AK3 (0.48) MAPTTP53RAB9ANPC1SMN1; SMN2
Hydrochloric Acid SCHEMBL6667512 0.83 EIF2AK3 (0.43) MAPTTP53RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383760-A1 BIARYLCARBOXAMIDE COMPOUNDS AS APOLIPOPROTEIN B INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-01-28 EP disclosed
WO-2002090347-A1 AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-11-14 WO disclosed