SCHEMBL6668516

SCHEMBL6668516

CCCN(C)n1ccnc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 1/20 0.37
CYP19A1 P11511 9/20 0.36
NFKB1 P19838 1/20 0.34
QPCT Q16769 1/20 0.34
HSD17B10 Q99714 1/20 0.34
QPCTL Q9NXS2 1/20 0.34
HTT P42858 1/20 0.34
CYP1A2 P05177 4/20 0.32
CYP2D6 P10635 4/20 0.32
CYP2C9 P11712 4/20 0.32
CYP2C19 P33261 4/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
CYP3A4 P08684 3/20 0.31
ALOX15 P16050 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28183020 0.88 TBXAS1 (0.43) TBXAS1CYP19A1NFKB1QPCTHSD17B10
SCHEMBL28182996 0.85
Water SCHEMBL27804544 0.83 CYP19A1 (0.38) TBXAS1CYP19A1NFKB1QPCTHSD17B10
SCHEMBL29175060 0.79 PRMT3 (0.37) CYP19A1NFKB1QPCTHSD17B10QPCTL
SCHEMBL29082466 0.73 TBXAS1 (0.44) TBXAS1CYP19A1NFKB1QPCTHSD17B10
SCHEMBL5132791 0.73 TBXAS1 (0.33) TBXAS1CYP19A1NFKB1QPCTHSD17B10
SCHEMBL4878051 0.73 NFKB1 (0.34) TBXAS1CYP19A1NFKB1QPCTHSD17B10
SCHEMBL4394208 0.72
SCHEMBL6398854 0.72 EGLN3 (0.40) TBXAS1CYP19A1
SCHEMBL4106428 0.71 GRIN2D (0.33) TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1359916-A4 IMIDAZOLYL DERIVATIVES AS CORTICOTROPIN RELEASING FACTOR INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2004-04-07 EP disclosed
EP-1359916-A1 IMIDAZOLYL DERIVATIVES AS CORTICOTROPIN RELEASING FACTOR INHIBITORS Bristol-Myers Squibb Company (US) 2003-11-12 EP disclosed
WO-2002058704-A1 IMIDAZOLYL DERIVATIVES AS CORTICOTROPIN RELEASING FACTOR INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2002-08-01 WO disclosed
WO-1993013075-A1 1-(ARYLALKYL-AMINOALKYL)IMIDAZOLE DERIVATIVES, PROCESSES OF PREPARATION AND USE AS THERAPEUTICAL AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed