SCHEMBL6668902

SCHEMBL6668902

CC(=O)Oc1ccc(C#Cc2cc3c(cc2C)OCCC3(C)C)s1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RARA P10276 4/20 0.38
RARB P10826 4/20 0.38
RARG P13631 4/20 0.38
RXRA P19793 2/20 0.37
HNF4A P41235 2/20 0.37
CYP26A1 O43174 1/20 0.33
CYP26B1 Q9NR63 1/20 0.33
AKR1B1 P15121 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9142284 0.81 RXRA (0.41) RARARARBRARGRXRAHNF4A
SCHEMBL8884872 0.81 CYP26A1 (0.42) RARARARBRARGRXRAHNF4A
SCHEMBL9137414 0.80 RXRA (0.39) RARARARBRARGRXRAHNF4A
SCHEMBL9139421 0.76 RXRA (0.37) RARARARBRARGRXRAHNF4A
SCHEMBL6664143 0.76 RXRA (0.37) RARARARBRARGRXRAHNF4A
SCHEMBL9817878 0.73 RXRA (0.44) RARARARBRARGRXRAHNF4A
SCHEMBL7817655 0.73 ACACB (0.32) RARARARBRARGRXRAHNF4A
SCHEMBL9136509 0.72 RARB (0.36) RARARARBRARGRXRAHNF4A
SCHEMBL10571276 0.71 RARA (0.46) RARARARBRARGRXRAHNF4A
SCHEMBL6664577 0.70 CYP26A1 (0.41) RARARARBRARGRXRAHNF4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0785782-B1 USE OF DISUBSTITUTED ACETYLENES BEARING HETEROAROMATIC AND HETEROBICYCLIC GROUPS HAVING RETINOID-LIKE ACTIVITY ALLERGAN INC (US) 2004-09-08 EP disclosed