SCHEMBL6670153

SCHEMBL6670153

O=C1NC(=O)/C(=C\c2cccc(Br)c2)N1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
MAPT P10636 2/20 0.67
KDM4E B2RXH2 1/20 0.67
BLM P54132 1/20 0.67
L3MBTL1 Q9Y468 1/20 0.67
CISD1 Q9NZ45 3/20 0.55
MAOA P21397 1/20 0.55
MAOB P27338 1/20 0.55
PIM1 P11309 1/20 0.55
PIM2 Q9P1W9 1/20 0.55
GSK3B P49841 5/20 0.51
CGAS Q8N884 1/20 0.51
HSD11B1 P28845 1/20 0.50
PNP P00491 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ALPI P09923 1/20 0.48
LMNA P02545 1/20 0.47
RAB9A P51151 1/20 0.47
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6670159 1.00 MEN1 (0.67) MEN1KMT2AMAPTKDM4EBLM
SCHEMBL8012399 0.80 MAPT (0.67) MEN1KMT2AMAPTKDM4EBLM
SCHEMBL15305605 0.80 MEN1 (0.67) MEN1KMT2AMAPTKDM4EBLM
SCHEMBL28813132 0.80 MEN1 (1.00) MEN1KMT2AMAPTKDM4EBLM
SCHEMBL8012401 0.80 MAPT (0.67) MEN1KMT2AMAPTKDM4EBLM
SCHEMBL29727412 0.79 LMNA (0.70) MEN1KMT2AMAPTKDM4EBLM
SCHEMBL28818211 0.79 LMNA (0.70) MEN1KMT2AMAPTKDM4EBLM
SCHEMBL14031533 0.78 GSK3B (0.67) MEN1KMT2AMAPTKDM4EBLM
SCHEMBL1358078 0.78 GSK3B (0.67) MEN1KMT2AMAPTKDM4EBLM
SCHEMBL1358077 0.78 GSK3B (0.67) MEN1KMT2AMAPTKDM4EBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040121965-A1 Method of treating resistant tumors WYETH HOLDINGS CORPORATION (US) 2004-06-24 US disclosed
WO-2004026293-A2 HEMIASTERLIN DERIVATIVES FOR TREATING RESISTANT TUMORS WYETH HOLDINGS CORPORATION (US) 2004-04-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040121965-A1 Method of treating resistant tumors SLC11A2, VHL, REN MEN1 40/4885KMT2A 1114/4885MAPT 4461/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.