SCHEMBL6670425

SCHEMBL6670425

O=C([C@@H]1Cc2ccccc2N1C(=O)CCC1Cc2ccccc2C12CCNCC2)N1CCOCC1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.42
HTR1A P08908 3/20 0.40
HTR7 P34969 3/20 0.40
LMNA P02545 1/20 0.40
AKT1 P31749 2/20 0.38
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6672515 0.84 AKT1 (0.40) AKT1
SCHEMBL6672242 0.84 AKT1 (0.40) AKT1
SCHEMBL6672759 0.82 DRD2 (0.46)
SCHEMBL6673179 0.79 POLB (0.42) HTR7LMNA
SCHEMBL6669410 0.74 MC4R (0.42)
SCHEMBL6397610 0.74 OPRL1 (0.47) TP53HTR1AHTR7OPRM1OPRL1
SCHEMBL6397606 0.74 OPRL1 (0.47) TP53HTR1AHTR7OPRM1OPRL1
Hydrochloric Acid SCHEMBL6396517 0.74 OPRL1 (0.46) TP53HTR1AHTR7OPRM1OPRL1
SCHEMBL6674849 0.73 NOTUM (0.38)
Hydrochloric Acid SCHEMBL6669828 0.71 HTR2A (0.36) LMNAOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1399432-A1 SPIROPIPERIDINE COMPOUNDS AS LIGANDS FOR ORL-1 RECEPTOR PFIZER INC. (US) 2004-03-24 EP disclosed
WO-2003000677-A1 SPIROPIPERIDINE COMPOUNDS AS LIGANDS FOR ORL-1 RECEPTOR PFIZER PHARMACEUTICALS INC. (JP) 2003-01-03 WO disclosed