SCHEMBL667137

SCHEMBL667137

CCCC(N(NC(=O)c1cccc(OC)c1C)C(=O)c1cc(C)cc(C)c1)C(C)(C)C

nearest known ligand 0.64

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.64
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
UTS2R Q9UKP6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29684635 1.00 ABCB1 (0.64) ABCB1TAS1R3TAS1R1UTS2R
SCHEMBL2682557 1.00 ABCB1 (0.64) ABCB1TAS1R3TAS1R1UTS2R
SCHEMBL2681881 1.00 ABCB1 (0.64) ABCB1TAS1R3TAS1R1UTS2R
SCHEMBL29727267 0.94 ABCB1 (0.62) ABCB1UTS2R
SCHEMBL668804 0.94 ABCB1 (0.62) ABCB1UTS2R
SCHEMBL667855 0.93 ABCB1 (0.54) ABCB1TAS1R3TAS1R1UTS2R
SCHEMBL29684814 0.93 ABCB1 (0.54) ABCB1TAS1R3TAS1R1UTS2R
SCHEMBL2681921 0.93 ABCB1 (0.54) ABCB1TAS1R3TAS1R1UTS2R
SCHEMBL3766257 0.93 ABCB1 (0.60) ABCB1
SCHEMBL668812 0.92 ABCB1 (0.66) ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3357904-B1 CHIRAL DIACHYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX PRECIGEN INC (US) 2022-07-06 EP claimed
US-20200270225-A1 Chiral Diacylhydrazine Ligands for Modulating the Expression of Exogenous Genes via an Ecdysone Receptor Complex INTREXON CORPORATION (US) 2020-08-27 US claimed
EP-3568474-A1 MODULATING EXPRESSION OF POLYPEPTIDES VIA NEW GENE SWITCH EXPRESSION SYSTEMS Intrexon Corporation (US) 2019-11-20 EP claimed
EP-3357904-A1 CHIRAL DIACHYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX Intrexon Corporation (US) 2018-08-08 EP claimed
WO-2018132494-A1 MODULATING EXPRESSION OF POLYPEPTIDES VIA NEW GENE SWITCH EXPRESSION SYSTEMS INTREXON CORPORATION (US) 2018-07-19 WO claimed
EP-2167458-B1 CHIRAL DIACYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX INTREXON CORP (US) 2018-03-14 EP claimed
US-9359289-B2 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORPORATION (US) 2016-06-07 US claimed
EP-2460786-B1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORP (US) 2016-01-13 EP claimed
US-20150240244-A1 BIOAVAILABLE DIACYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT (GB) 2015-08-27 US claimed
US-9102648-B1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORPORATION (US) 2015-08-11 US claimed
US-20140045903-A1 Bioavailable Diacylhydrazine Ligands for Modulating the Expression of Exogenous Genes via an Ecdysone Receptor Complex INTREXON CORPORATION (US) 2014-02-13 US claimed
US-20130040389-A1 Bioavailable Diacylhydrazine Ligands for Modulating the Expression of Exogenous Genes via an Ecdysone Receptor Complex Intrexon Coporation (US) 2013-02-14 US claimed
EP-2460786-A1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex Intrexon Corporation (US) 2012-06-06 EP claimed
US-20120046322-A1 Bioavailable Diacylhydrazine Ligands for Modulating the Expression of Exogenous Genes via an Ecdysone Receptor Complex INTREXON CORPORATION (US) 2012-02-23 US claimed
US-20080064741-A1 BIOAVAILABLE DIACYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX RHEOGENE, INC. 2008-03-13 US claimed
EP-1601642-A4 BIOAVAILABLE DIACYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX RHEOGENE INC (US) 2007-04-11 EP claimed
US-20060020146-A1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex RHEOGENE, INC. 2006-01-26 US claimed
EP-1601642-A2 BIOAVAILABLE DIACYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX RheoGene, Inc. (US) 2005-12-07 EP claimed
WO-2004078924-A2 BIOAVAILABLE DIACYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX RHEOGENE, INC. (US) 2004-09-16 WO claimed
US-20260098063-A1 HUMAN PAPILLOMAVIRUS VACCINES AND USES OF THE SAME PRECIGEN INC (US) 2026-04-09 US disclosed
US-20260035432-A1 ROR-1 SPECIFIC CHIMERIC ANTIGEN RECEPTORS AND USES THEREOF PRECIGEN, INC. (US) 2026-02-05 US disclosed
US-12404306-B2 Human papillomavirus vaccines and uses of the same PRECIGEN, INC. (US) 2025-09-02 US disclosed
US-20250223320-A1 HEPATITIS B VACCINES AND USES OF THE SAME PRECIGEN, INC. (US) 2025-07-10 US disclosed
US-12275772-B2 ROR-1 specific chimeric antigen receptors and uses thereof PRECIGEN, INC. (US) 2025-04-15 US disclosed
US-12234261-B2 Hepatitis B vaccines and uses of the same PRECIGEN, INC. (US) 2025-02-25 US disclosed
US-20240368305-A1 MUC16 SPECIFIC CHIMERIC ANTIGEN RECEPTORS AND USES THEREOF PRECIGEN, INC. (US) 2024-11-07 US disclosed
US-20240263183-A1 MODULATING EXPRESSION OF POLYPEPTIDES VIA NEW GENE SWITCH EXPRESSION SYSTEMS PRECIGEN, INC. (US) 2024-08-08 US disclosed
EP-4382913-A2 MODULATING EXPRESSION OF POLYPEPTIDES VIA NEW GENE SWITCH EXPRESSION SYSTEMS Precigen, Inc. (US) 2024-06-12 EP disclosed
US-20240173396-A1 Human Papilloma Virus Vaccines and Uses of the Same for HPV Associated Diseases BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT (GB) 2024-05-30 US disclosed
US-11981746-B2 MUC16 specific chimeric antigen receptors and uses thereof PRECIGEN, INC. (US) 2024-05-14 US disclosed
US-11976134-B2 MUC16 specific chimeric antigen receptors and uses thereof PRECIGEN, INC. (US) 2024-05-07 US disclosed
US-11946054-B2 Modulating expression of polypeptides via new gene switch expression systems PRECIGEN, INC. (US) 2024-04-02 US disclosed
EP-4274898-A2 CHIMERIC RECEPTOR THERAPY Precigen, Inc. (US) 2023-11-15 EP disclosed
EP-4251278-A1 HUMAN PAPILLOMA VIRUS VACCINES AND USES OF THE SAME FOR HPV ASSOCIATED DISEASES Precigen, Inc. (US) 2023-10-04 EP disclosed
US-20230279057-A1 HEPATITIS B VACCINES AND USES OF THE SAME PRECIGEN, INC. (US) 2023-09-07 US disclosed
US-11692194-B2 Modulating expression of polypeptides via new gene switch expression systems PRECIGEN, INC. (US) 2023-07-04 US disclosed
US-11608362-B2 Hepatitis B vaccines and uses of the same PRECIGEN, INC. (US) 2023-03-21 US disclosed
WO-2022150732-A2 CHIMERIC RECEPTOR THERAPY PRECIGEN, INC. (US) 2022-07-14 WO disclosed
US-20220220187-A1 CHIMERIC RECEPTOR THERAPY BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT (GB) 2022-07-14 US disclosed
EP-3357904-B1 CHIRAL DIACHYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX PRECIGEN INC (US) 2022-07-06 EP disclosed
EP-3357904-B1 CHIRAL DIACHYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX PRECIGEN INC (US) 2022-07-06 EP disclosed
WO-2022115470-A1 HUMAN PAPILLOMA VIRUS VACCINES AND USES OF THE SAME FOR HPV ASSOCIATED DISEASES PRECIGEN, INC. (US) 2022-06-02 WO disclosed
US-20220153866-A1 MUC16 SPECIFIC CHIMERIC ANTIGEN RECEPTORS AND USES THEREOF PRECIGEN, INC. (US) 2022-05-19 US disclosed
US-20220153867-A1 MUC16 SPECIFIC CHIMERIC ANTIGEN RECEPTORS AND USES THEREOF PRECIGEN, INC. (US) 2022-05-19 US disclosed
US-11319380-B2 MUC16 specific chimeric antigen receptors and uses thereof PRECIGEN, INC. (US) 2022-05-03 US disclosed
US-20210177902-A1 ROR-1 SPECIFIC CHIMERIC ANTIGEN RECEPTORS AND USES THEREOF BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT (GB) 2021-06-17 US disclosed
EP-3802615-A2 MUC16 SPECIFIC CHIMERIC ANTIGEN RECEPTORS AND USES THEREOF Precigen, Inc. (US) 2021-04-14 EP disclosed
US-20210024586-A1 HUMAN PAPILLOMAVIRUS VACCINES AND USES OF THE SAME PRECIGEN, INC. (US) 2021-01-28 US disclosed
US-20210015911-A1 HEPATITIS B VACCINES AND USES OF THE SAME PRECIGEN, INC. (US) 2021-01-21 US disclosed
EP-3762022-A1 HUMAN PAPILLOMAVIRUS VACCINES AND USES OF THE SAME Precigen, Inc. (US) 2021-01-13 EP disclosed
EP-3762010-A1 HEPATITIS B VACCINES AND USES OF THE SAME Precigen, Inc. (US) 2021-01-13 EP disclosed
US-20200283778-A1 MODULATING EXPRESSION OF POLYPEPTIDES VIA NEW GENE SWITCH EXPRESSION SYSTEMS PRECIGEN, INC. (US) 2020-09-10 US disclosed
EP-3568474-A1 MODULATING EXPRESSION OF POLYPEPTIDES VIA NEW GENE SWITCH EXPRESSION SYSTEMS Intrexon Corporation (US) 2019-11-20 EP disclosed
WO-2019173465-A1 HUMAN PAPILLOMAVIRUS VACCINES AND USES OF THE SAME INTREXON CORPORATION (US) 2019-09-12 WO disclosed
WO-2019173463-A1 HEPATITIS B VACCINES AND USES OF THE SAME INTREXON CORPORATION (US) 2019-09-12 WO disclosed
US-20180291384-A1 MODULATING EXPRESSION OF POLYPEPTIDES VIA NEW GENE SWITCH EXPRESSION SYSTEMS BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT (GB) 2018-10-11 US disclosed
EP-3357904-A1 CHIRAL DIACHYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX Intrexon Corporation (US) 2018-08-08 EP disclosed
EP-3357904-A1 CHIRAL DIACHYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX Intrexon Corporation (US) 2018-08-08 EP disclosed
WO-2018132494-A1 MODULATING EXPRESSION OF POLYPEPTIDES VIA NEW GENE SWITCH EXPRESSION SYSTEMS INTREXON CORPORATION (US) 2018-07-19 WO disclosed
EP-2167458-B1 CHIRAL DIACYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX INTREXON CORP (US) 2018-03-14 EP disclosed
EP-2167458-B1 CHIRAL DIACYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX INTREXON CORP (US) 2018-03-14 EP disclosed
EP-2463269-B1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORP (US) 2016-09-28 EP disclosed
EP-2460786-B1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORP (US) 2016-01-13 EP disclosed
EP-2463269-A1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex Intrexon Corporation (US) 2012-06-13 EP disclosed
EP-2460786-A1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex Intrexon Corporation (US) 2012-06-06 EP disclosed
EP-2460786-A1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex Intrexon Corporation (US) 2012-06-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120046322-A1 Bioavailable Diacylhydrazine Ligands for Modulating the Expression of Exogenous Genes via an Ecdysone Receptor Complex NR2E3, NR5A1, NR5A2 ABCB1 1365/4885TAS1R3 2234/4885TAS1R1 2333/4885
US-20260035432-A1 ROR-1 SPECIFIC CHIMERIC ANTIGEN RECEPTORS AND USES THEREOF RORB, ICOS, RORC ABCB1 2759/4885TAS1R3 3559/4885TAS1R1 3066/4885
US-20260098063-A1 HUMAN PAPILLOMAVIRUS VACCINES AND USES OF THE SAME ANKRD54, POTEE, ANKK1 ABCB1 4133/4885TAS1R3 1710/4885TAS1R1 2369/4885
US-20080064741-A1 BIOAVAILABLE DIACYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX NR2E3, NR5A1, NR5A2 ABCB1 1365/4885TAS1R3 2234/4885TAS1R1 2333/4885
US-20130040389-A1 Bioavailable Diacylhydrazine Ligands for Modulating the Expression of Exogenous Genes via an Ecdysone Receptor Complex NR2E3, NR5A1, NR5A2 ABCB1 1365/4885TAS1R3 2234/4885TAS1R1 2333/4885
US-20220220187-A1 CHIMERIC RECEPTOR THERAPY HAVCR2, PTPN6, PTPN18 ABCB1 1438/4885TAS1R3 2987/4885TAS1R1 2984/4885
US-20060020146-A1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex NR2E3, NR5A1, NR5A2 ABCB1 1365/4885TAS1R3 2234/4885TAS1R1 2333/4885
US-20200270225-A1 Chiral Diacylhydrazine Ligands for Modulating the Expression of Exogenous Genes via an Ecdysone Receptor Complex NR2E3, CRYZ, TCF12 ABCB1 692/4885TAS1R3 3889/4885TAS1R1 4166/4885
US-20140045903-A1 Bioavailable Diacylhydrazine Ligands for Modulating the Expression of Exogenous Genes via an Ecdysone Receptor Complex NR2E3, NR2C2, NR5A2 ABCB1 1302/4885TAS1R3 2240/4885TAS1R1 2323/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.