SCHEMBL6672302

SCHEMBL6672302

O=C(O)Cc1c(-c2ccccc2)[nH]c2ncccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.49
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
FNTA P49354 6/20 0.47
FNTB P49356 6/20 0.47
CCNB2 O95067 1/20 0.47
CDK1 P06493 1/20 0.47
CCNB1 P14635 1/20 0.47
GSK3A P49840 1/20 0.47
GSK3B P49841 1/20 0.47
CCNB3 Q8WWL7 1/20 0.47
PPARG P37231 2/20 0.46
AURKA O14965 1/20 0.44
PARP1 P09874 1/20 0.44
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1780538 0.89 CNR1 (0.47) CNR1ADORA2AADORA1FNTAFNTB
SCHEMBL1778459 0.84 CNR1 (0.44) CNR1ADORA2AADORA1FNTAFNTB
SCHEMBL1778871 0.82 GSK3A (0.65) FNTAFNTBCCNB2CDK1CCNB1
SCHEMBL857278 0.82 CCNB2 (0.68) CNR1ADORA2AADORA1FNTAFNTB
SCHEMBL16497186 0.81 KDM4E (0.48) AURKAPARP1KDM4EALDH1A1GAA
SCHEMBL1778456 0.80 MTNR1A (0.66) KDM4EALDH1A1
SCHEMBL29868708 0.80 MTNR1A (0.66) KDM4EALDH1A1
SCHEMBL8140328 0.79 HTR6 (0.64) CNR1ADORA2AADORA1CCNB2CDK1
SCHEMBL1778446 0.78 HTR6 (0.49) CNR1ADORA2AADORA1FNTAFNTB
SCHEMBL1777136 0.78 CLK1 (0.49) CNR1ADORA2AADORA1FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1324985-A4 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 2004-10-06 EP disclosed
EP-1324985-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2003-07-09 EP disclosed
WO-2002028831-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2002-04-11 WO disclosed