SCHEMBL6672392

SCHEMBL6672392

C#CCOC[C@H]1O[C@@H](n2cnc3c(NC4CC4(C)C)ncnc32)[C@H](O)[C@@H]1O

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.61
ADORA1 P30542 8/20 0.59
TAS1R3 Q7RTX0 1/20 0.53
TAS1R1 Q7RTX1 1/20 0.53
TSHR P16473 2/20 0.52
ADORA2A P29274 2/20 0.52
ADORA2B P29275 2/20 0.52
PMP22 Q01453 1/20 0.52
GAA P10253 1/20 0.52
HTT P42858 1/20 0.52
SIGMAR1 Q99720 1/20 0.52
SLC29A1 Q99808 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
TP53 P04637 1/20 0.52
NFKB1 P19838 1/20 0.52
HIF1A Q16665 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6673454 0.88 ADORA3 (0.73) ADORA3ADORA1TAS1R3TAS1R1TSHR
SCHEMBL6685672 0.85 ADORA3 (0.71) ADORA3ADORA1TAS1R3TAS1R1TSHR
SCHEMBL6685682 0.85 ADORA3 (0.71) ADORA3ADORA1TAS1R3TAS1R1TSHR
SCHEMBL6671330 0.84 ADORA1 (0.71) ADORA3ADORA1ADORA2AADORA2BPMP22
SCHEMBL6670773 0.84 ADORA3 (0.73) ADORA3ADORA1TAS1R3TAS1R1TSHR
SCHEMBL6258690 0.82 AHCY (0.61) ADORA3ADORA1TSHRADORA2AADORA2B
SCHEMBL6671096 0.81 ADORA3 (0.55) ADORA3ADORA1TAS1R3TAS1R1TSHR
SCHEMBL6671101 0.81 ADORA3 (0.55) ADORA3ADORA1TAS1R3TAS1R1TSHR
SCHEMBL6670771 0.81 ADORA3 (0.68) ADORA3ADORA1TAS1R3TAS1R1ADORA2A
SCHEMBL6670776 0.81 ADORA3 (0.68) ADORA3ADORA1TAS1R3TAS1R1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004026890-A1 ACETYLENE COMPOUNDS GLAXO GROUP LIMITED (GB) 2004-04-01 WO claimed
WO-2004026890-A1 ACETYLENE COMPOUNDS GLAXO GROUP LIMITED (GB) 2004-04-01 WO disclosed