SCHEMBL6673085

SCHEMBL6673085

O=C(OCCCCc1ccccc1)c1cccnc1N1CCN(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 9/20 0.54
SLC6A3 Q01959 7/20 0.54
HTR2A P28223 7/20 0.54
DRD5 P21918 6/20 0.54
DRD4 P21917 6/20 0.54
HTR7 P34969 6/20 0.54
HRH1 P35367 5/20 0.54
OPRM1 P35372 5/20 0.54
CACNA1F O60840 4/20 0.54
HRH2 P25021 4/20 0.54
ADRA1D P25100 4/20 0.54
ADRA1A P35348 4/20 0.54
ADRA1B P35368 4/20 0.54
HTR6 P50406 4/20 0.54
CACNA1D Q01668 4/20 0.54
CACNA1S Q13698 4/20 0.54
CACNA1C Q13936 4/20 0.54
OPRK1 P41145 4/20 0.54
DRD1 P21728 4/20 0.54
HTR2C P28335 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6672090 0.99 DRD3 (0.54) DRD3SLC6A3HTR2ADRD5DRD4
SCHEMBL7772096 0.95 SLC6A3 (0.58) DRD3SLC6A3HTR2ADRD5DRD4
SCHEMBL7773593 0.90 DRD3 (0.51) DRD3SLC6A3HTR2ADRD5DRD4
SCHEMBL7771969 0.87 LMNA (0.52) DRD3SLC6A3HTR2ADRD5DRD4
Hydrochloric Acid SCHEMBL7794427 0.86 LMNA (0.51) DRD3SLC6A3HTR2ADRD5DRD4
SCHEMBL7794410 0.86 LMNA (0.52) DRD3SLC6A3HTR2ADRD5DRD4
SCHEMBL6673075 0.86 LMNA (0.53) DRD3SLC6A3HTR2ADRD5DRD4
Hydrochloric Acid SCHEMBL7794406 0.85 LMNA (0.51) DRD3SLC6A3HTR2ADRD5DRD4
Hydrochloric Acid SCHEMBL6672087 0.85 LMNA (0.52) DRD3SLC6A3HTR2ADRD5DRD4
SCHEMBL6672744 0.85 DRD3 (0.46) DRD3SLC6A3HTR2ADRD5DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658910-A TREATING MENTAL DISORDERS PHARMACIA AB (SE) 1997-08-19 US claimed
EP-1120410-B1 Nicotinic acid esters useful as CNS agents and having affinity for 5-HT receptors BIOVITRUM AB (SE) 2004-10-06 EP disclosed
EP-1120410-A1 Nicotinic acid esters useful as CNS agents and having affinity for 5-HT receptors Pharmacia AB (SE) 2001-08-01 EP disclosed
US-5658910-A TREATING MENTAL DISORDERS PHARMACIA AB (SE) 1997-08-19 US disclosed