SCHEMBL6673645

SCHEMBL6673645

NC(=O)c1ccccc1CC(F)(F)C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
METAP2 P50579 1/20 0.40
BCAT2 O15382 1/20 0.39
PDK2 Q15119 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
AURKB Q96GD4 1/20 0.37
MAOB P27338 1/20 0.37
GAA P10253 2/20 0.36
CTNNB1 P35222 1/20 0.36
LMNA P02545 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363265 0.85 KDM4E (0.45) KDM4EALDH1A1MAPTHPGDTSHR
Hydrochloric Acid SCHEMBL28047477 0.84 KDM4E (0.44) KDM4EALDH1A1MAPTHPGDTSHR
Hydrochloric Acid SCHEMBL27491870 0.84 KDM4E (0.44) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL13508575 0.78 KDM4E (0.45) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL29818200 0.78 KDM4E (0.45) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL21590341 0.76 KDM4E (0.44) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL31628129 0.75 CES1 (0.52) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL28316789 0.75 ALDH1A1 (0.42) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL3828592 0.75 KDM4E (0.50) KDM4EALDH1A1MAPTHPGDTSHR
SCHEMBL29713752 0.75 HDAC1 (0.36) ALDH1A1MEN1KMT2AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1461317-A2 PROCESS FOR PREPARING HYDROXYPYRROLIDINYL ETHYLAMINE COMPOUNDS USEFUL AS KAPPA AGONISTS Pfizer Products Inc. (US) 2004-09-29 EP disclosed
WO-2002088082-A2 PROCESS FOR PREPARING HYDROXYPYRROLIDINYL ETHYLAMINE COMPOUNDS USEFUL AS KAPPA AGONISTS PFIZER PRODUCTS INC. (US) 2002-11-07 WO disclosed