SCHEMBL6673750

SCHEMBL6673750

C[SiH](C)OC(c1ccccc1C(=O)O)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
KMT2A Q03164 4/20 0.41
TDP1 Q9NUW8 2/20 0.41
GAA P10253 1/20 0.41
ALOX15 P16050 2/20 0.39
KDM4E B2RXH2 5/20 0.38
HPGD P15428 3/20 0.38
HSD17B10 Q99714 3/20 0.38
MAPT P10636 2/20 0.38
HDAC8 Q9BY41 1/20 0.38
HMGB1 P09429 2/20 0.37
NAPRT Q6XQN6 2/20 0.37
ESR1 P03372 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
TSHR P16473 1/20 0.37
GGT1 P19440 1/20 0.37
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
BLM P54132 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10349585 0.85 ALDH1A1 (0.39) ALDH1A1KMT2ATDP1GAAALOX15
SCHEMBL4609062 0.81 PDK2 (0.34) ALDH1A1TDP1TSHRHTTRECQL
SCHEMBL7045747 0.80 TRPM8 (0.36) CA1CA2CA9
SCHEMBL1465848 0.75
SCHEMBL4279554 0.74 PDE4A (0.32)
SCHEMBL2082916 0.73 LMNA (0.38) ALDH1A1KMT2ATDP1GAAHPGD
SCHEMBL4298018 0.73 APOBEC3G (0.32)
SCHEMBL6671659 0.72 NR1H4 (0.42) ALDH1A1KMT2AHPGDTSHRCA12
SCHEMBL27433644 0.71 ALDH1A1 (0.50) ALDH1A1KMT2ATDP1GAAALOX15
SCHEMBL4609578 0.70 PDE2A (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0751144-B1 Novel anthracycline prodrugs, method for preparation as well as their use in selective chemotherapy PHARMACHEMIE BV (NL) 2004-10-06 EP disclosed
US-5710135-A ENZYMATICALLY CLEAVABLE; ANTITUMOR AGENTS PHARMACHEMIE B.V. (NL) 1998-01-20 US disclosed
EP-0751144-A1 Novel anthracycline prodrugs, method for preparation as well as their use in selective chemotherapy PHARMACHEMIE B.V. (NL) 1997-01-02 EP disclosed