SCHEMBL6674384

SCHEMBL6674384

Cc1c(CN(C)C(=O)OC(C)(C)C)cccc1[N+](=O)[O-]

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.45
TSHR P16473 2/20 0.43
ALDH1A1 P00352 2/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
NR1D1 P20393 1/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6676029 0.88 TDP1 (0.46) TDP1TSHRALDH1A1HTTSMN1; SMN2
SCHEMBL2061458 0.88 ALDH1A1 (0.49) ALDH1A1HTTBCHEACHE
SCHEMBL27274797 0.87 GPR35 (0.45) ALDH1A1HTTNR1D1BCHEACHE
SCHEMBL30658955 0.87 GPR35 (0.45) ALDH1A1HTTNR1D1BCHEACHE
SCHEMBL24492402 0.86 RIPK1 (0.44) ALDH1A1HTTNR1D1BCHEACHE
SCHEMBL29465818 0.86 RIPK1 (0.44) ALDH1A1HTTNR1D1BCHEACHE
SCHEMBL4613668 0.80 ALDH1A1 (0.38) ALDH1A1HTTNR1D1BCHEACHE
SCHEMBL7647352 0.79 ALDH1A1 (0.48) TSHRALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL30408067 0.79 ALDH1A1 (0.48) TSHRALDH1A1HTTSMN1; SMN2NPC1
SCHEMBL30696948 0.79 RIPK1 (0.41) ALDH1A1HTTNR1D1BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
CN-1075808-C Aniline derivatives having nitric oxide synthase inhibitory activity CHUGAI PHARMACEUTICAL CO LTD (JP) 2001-12-05 CN disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed