SCHEMBL6674484

SCHEMBL6674484

CCN=C(N)Nc1cccc(C(C)N)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.40
GRIN2D O15399 5/20 0.40
GRIN3B O60391 5/20 0.40
GRIN1 Q05586 5/20 0.40
GRIN2A Q12879 5/20 0.40
GRIN2B Q13224 5/20 0.40
GRIN2C Q14957 5/20 0.40
GRIN3A Q8TCU5 5/20 0.40
CACNA1C Q13936 1/20 0.40
SCN5A Q14524 1/20 0.40
PTGIR P43119 2/20 0.36
CXCR4 P61073 2/20 0.34
NOS1 P29475 2/20 0.34
MEN1 O00255 1/20 0.34
PABPC1 P11940 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
EBP Q15125 1/20 0.34
TMEM97 Q5BJF2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6675375 0.99 SIGMAR1 (0.40) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6678288 0.82 PTGIR (0.40) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6676424 0.77 CACNA1C (0.48) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL6675369 0.75 CACNA1C (0.47) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6680201 0.74 CACNA1C (0.46) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL6675374 0.73 ALDH1A1 (0.40) SIGMAR1KMT2AALDH1A1MAPTHSD17B10
Hydrochloric Acid SCHEMBL6679115 0.73 CACNA1C (0.45) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6675327 0.73 CACNA1C (0.45) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
Hydrochloric Acid SCHEMBL6679167 0.72 CACNA1C (0.44) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL6679082 0.70 SIGMAR1 (0.52) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP claimed