SCHEMBL6674574

SCHEMBL6674574

CC(N)(CCc1ccccc1)c1ccc(O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.48
ESR2 Q92731 6/20 0.48
CYP3A4 P08684 4/20 0.48
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
SLC6A2 P23975 2/20 0.41
TAAR1 Q96RJ0 1/20 0.41
BLM P54132 1/20 0.41
KIF11 P52732 1/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
LMNA P02545 1/20 0.41
TYR P14679 1/20 0.41
AR P10275 1/20 0.41
TSHR P16473 1/20 0.41
SLC6A4 P31645 1/20 0.41
HTR6 P50406 1/20 0.41
ESRRG P62508 1/20 0.41
SLC6A3 Q01959 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865764 0.82 SLC6A2 (0.53) ESR1ESR2CYP3A4ALDH1A1SLC6A2
SCHEMBL311387 0.82 ESR1 (0.56) ESR1ESR2CYP3A4ALDH1A1MEN1
SCHEMBL8976239 0.81 ESR1 (0.56) ESR1ESR2CYP3A4ALDH1A1MEN1
Hydrochloric Acid SCHEMBL8866021 0.81 SLC6A2 (0.52) ESR1ESR2CYP3A4ALDH1A1SLC6A2
SCHEMBL20492109 0.77 KIF11 (0.53) ESR1ESR2CYP3A4ALDH1A1SLC6A2
SCHEMBL28674136 0.76 ESR1 (0.48) ESR1ESR2CYP3A4ALDH1A1MEN1
SCHEMBL10656617 0.75 ESR1 (0.58) ESR1ESR2CYP3A4ALDH1A1SLC6A2
SCHEMBL8866151 0.75 BLM (0.56) ESR1ESR2CYP3A4ALDH1A1SLC6A2
SCHEMBL7837799 0.75 ESR1 (0.56) ESR1ESR2CYP3A4ALDH1A1MEN1
Hydrochloric Acid SCHEMBL8865821 0.74 BLM (0.54) ESR1ESR2CYP3A4ALDH1A1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1305852-C Diaryl ethers as opioid receptor antagonists LILLY CO ELI (US) 2007-03-21 CN disclosed
CN-1681498-A Diaryl ethers as opioid receptor antagonist LILLY CO ELI (US) 2005-10-12 CN disclosed
WO-2004026305-A9 DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST LILLY CO ELI (US) 2004-05-13 WO disclosed