SCHEMBL6674653

SCHEMBL6674653

O=C(O)C(=O)Cc1cc2ccccc2s1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.58
ASIC3 Q9UHC3 1/20 0.53
LOXL2 Q9Y4K0 1/20 0.53
BCL2L1 Q07817 1/20 0.51
AGXT P21549 1/20 0.49
ADRB2 P07550 1/20 0.49
GLS O94925 2/20 0.48
DRD2 P14416 1/20 0.48
DRD4 P21917 1/20 0.48
DRD3 P35462 1/20 0.48
KDM4C Q9H3R0 1/20 0.48
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47
CA5A P35218 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
CA5B Q9Y2D0 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29534459 0.86 CYP2A6 (0.61) CYP2A6ASIC3LOXL2BCL2L1AGXT
SCHEMBL631264 0.86 CYP2A6 (0.61) CYP2A6ASIC3LOXL2BCL2L1AGXT
SCHEMBL28666644 0.81 CYP2A6 (0.56) CYP2A6ASIC3LOXL2BCL2L1AGXT
SCHEMBL29861035 0.81 CYP2A6 (0.56) CYP2A6ASIC3LOXL2BCL2L1AGXT
SCHEMBL1029348 0.81 CYP2A6 (0.59) CYP2A6ASIC3LOXL2BCL2L1AGXT
SCHEMBL1260041 0.81 CYP2A6 (0.59) CYP2A6ASIC3LOXL2BCL2L1AGXT
SCHEMBL11215245 0.81 CYP2A6 (0.59) CYP2A6ASIC3LOXL2BCL2L1AGXT
SCHEMBL31356469 0.81 CYP2A6 (0.59) CYP2A6ASIC3LOXL2BCL2L1AGXT
SCHEMBL11221971 0.79 CYP2A6 (0.58) CYP2A6ASIC3LOXL2BCL2L1AGXT
SCHEMBL7140216 0.79 RAB9A (0.49) CYP2A6ASIC3LOXL2AGXTADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040121965-A1 Method of treating resistant tumors WYETH HOLDINGS CORPORATION (US) 2004-06-24 US disclosed
WO-2004026293-A2 HEMIASTERLIN DERIVATIVES FOR TREATING RESISTANT TUMORS WYETH HOLDINGS CORPORATION (US) 2004-04-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040121965-A1 Method of treating resistant tumors SLC11A2, VHL, REN CYP2A6 2950/4885ASIC3 2801/4885LOXL2 758/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.