SCHEMBL6675259

SCHEMBL6675259

CN(C(=O)OC(C)(C)C)[C@H](C(=O)O)C(C)(C)c1ccc(C(=O)OC(C)(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
SLC7A5 Q01650 1/20 0.37
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
ALOX15 P16050 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34
MMP13 P45452 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
TDP1 Q9NUW8 2/20 0.33
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6675257 1.00 CA12 (0.39) CA12CA1CA2CA9CA14
SCHEMBL6810467 0.87 NOTUM (0.38) CA12CA1CA2CA9CA14
SCHEMBL22069882 0.86 ESR1 (0.36) MMP13HDAC3HDAC1HDAC2NCOR2
SCHEMBL20732299 0.86 ESR1 (0.36) MMP13HDAC3HDAC1HDAC2NCOR2
SCHEMBL58396 0.86 MMP13 (0.40) CYP1A2CYP2D6CYP2C19ALOX15MMP13
SCHEMBL88460 0.86 MMP13 (0.40) CYP1A2CYP2D6CYP2C19ALOX15MMP13
SCHEMBL5981030 0.86 MMP13 (0.40) CYP1A2CYP2D6CYP2C19ALOX15MMP13
SCHEMBL16183160 0.85 KIF11 (0.37) SLC7A5MMP13HDAC3HDAC1HDAC2
SCHEMBL16176598 0.85 AAK1 (0.40) CYP2D6CYP2C19MMP13TDP1MAPT
SCHEMBL20723962 0.85 AAK1 (0.35) SLC7A5MMP13MAPTALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040121965-A1 Method of treating resistant tumors WYETH HOLDINGS CORPORATION (US) 2004-06-24 US disclosed
WO-2004026293-A2 HEMIASTERLIN DERIVATIVES FOR TREATING RESISTANT TUMORS WYETH HOLDINGS CORPORATION (US) 2004-04-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040121965-A1 Method of treating resistant tumors SLC11A2, VHL, REN CA12 34/4885CA1 121/4885CA2 32/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.