SCHEMBL6675322

SCHEMBL6675322

O=C1c2ccccc2C(=O)N1Cc1cc([N+](=O)[O-])ccc1O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.59
LMNA P02545 1/20 0.59
CA12 O43570 2/20 0.56
CA1 P00915 2/20 0.56
CA2 P00918 2/20 0.56
CA9 Q16790 2/20 0.56
HSPD1 P10809 1/20 0.55
HSPE1 P61604 1/20 0.55
CTSB P07858 1/20 0.53
NOX4 Q9NPH5 1/20 0.52
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
RXFP1 Q9HBX9 1/20 0.50
CASP6 P55212 2/20 0.49
CASP1 P29466 1/20 0.49
CASP3 P42574 1/20 0.49
CASP4 P49662 1/20 0.49
CASP7 P55210 1/20 0.49
CASP9 P55211 1/20 0.49
CASP8 Q14790 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18231270 0.82 CA12 (0.49) KDM4ELMNACA12CA1CA2
SCHEMBL13172450 0.81 ALOX5 (0.48) KDM4ELMNACA12CA1CA2
SCHEMBL31455961 0.81 ALOX5 (0.48) KDM4ELMNACA12CA1CA2
SCHEMBL6675911 0.80 RXFP1 (0.62) KDM4ECA12CA1CA2CA9
SCHEMBL1832812 0.79 CA12 (0.60) LMNACA12CA1CA2CA9
SCHEMBL2049541 0.78 ALDH1A1 (0.73) CA12CA1CA2CA9MEN1
SCHEMBL31687464 0.78 ALDH1A1 (0.73) CA12CA1CA2CA9MEN1
SCHEMBL6679920 0.78 ALDH1A1 (0.52) LMNACA12CA1CA2CA9
SCHEMBL6841652 0.78 ALDH1A1 (0.57) CA12CA1CA2CA9HSPD1
SCHEMBL16241634 0.77 ALDH1A1 (0.48) KDM4ELMNACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed