SCHEMBL6675592

SCHEMBL6675592

COC(=O)C(CNC(=O)OC(C)(C)C)c1ccc(NC(N)=N[N+](=O)[O-])cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
PRMT1 Q99873 1/20 0.36
PTPN11 Q06124 1/20 0.35
AAK1 Q2M2I8 1/20 0.35
SYK P43405 1/20 0.34
MAPT P10636 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
LDHA P00338 1/20 0.33
LDHB P07195 1/20 0.33
CYP17A1 P05093 1/20 0.33
XBP1 P17861 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
NAMPT P43490 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6676230 0.91 PTPN11 (0.38) CA1CA2PRMT1PTPN11AAK1
SCHEMBL6680652 0.82 ALDH1A1 (0.40) CA1CA2PTPN11AAK1SYK
SCHEMBL6675651 0.82 GRIN2D (0.38) LDHALDHBGRIN2DGRIN3BGRIN1
SCHEMBL7247922 0.81 PTPN11 (0.38) CA1CA2PRMT1PTPN11AAK1
Hydrochloric Acid SCHEMBL6681329 0.81 GRIN2D (0.37) LDHALDHBGRIN2DGRIN3BGRIN1
SCHEMBL6676314 0.80 NAMPT (0.51) CA1CA2PRMT1PTPN11MAPT
SCHEMBL6675373 0.80 NPC1 (0.46) MAPTNPSR1KDM4E
SCHEMBL6677827 0.78 NAMPT (0.53) CA1CA2PRMT1PTPN11MAPT
SCHEMBL6680783 0.78 CA1 (0.40) CA1CA2PRMT1PTPN11CYP17A1
SCHEMBL6680756 0.78 ITGB3 (0.48) CA1CA2NPSR1GSTP1GSTM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed