SCHEMBL6680652

SCHEMBL6680652

COC(=O)C(CNC(=O)OC(C)(C)C)c1ccc(NC(N)=S)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
GAA P10253 2/20 0.40
PTPN11 Q06124 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
MAPKAPK2 P49137 4/20 0.39
AAK1 Q2M2I8 1/20 0.39
SYK P43405 1/20 0.38
LDHA P00338 1/20 0.37
LDHB P07195 1/20 0.37
CYP17A1 P05093 1/20 0.37
NAMPT P43490 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
MAPT P10636 3/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6679064 0.83 AAK1 (0.42) CA1CA2AAK1SYKESR1
SCHEMBL6675592 0.82 CA1 (0.37) PTPN11CA1CA2AAK1SYK
SCHEMBL2796410 0.81 L3MBTL1 (0.47) GAAAAK1SYKESR1ESR2
SCHEMBL31724105 0.81 ESR1 (0.45) GAACA1CA2AAK1SYK
SCHEMBL31724161 0.80 NPSR1 (0.43) ALDH1A1CA1CA2SYKESR1
SCHEMBL31389109 0.80 CTSS (0.43) ALDH1A1GAAAAK1SYKLDHA
SCHEMBL191176 0.80 L3MBTL1 (0.50) ALDH1A1GAASYKESR1ESR2
SCHEMBL31724221 0.80 SERPINE1 (0.44) GAACA1CA2AAK1SYK
SCHEMBL31724101 0.80 AAK1 (0.47) ALDH1A1AAK1SYKESR1ESR2
SCHEMBL6531538 0.80 SYK (0.52) SYKMAPTKMT2ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed