SCHEMBL6675978

SCHEMBL6675978

Cn1cc(N2Cc3cccc(-c4ccc(C(F)(F)F)cc4)c3C2=O)cc1OC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
RAB9A P51151 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
BACE1 P56817 1/20 0.38
POLB P06746 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ESR1 P03372 1/20 0.37
NR4A1 P22736 1/20 0.37
APEX1 P27695 1/20 0.37
PTPN7 P35236 1/20 0.37
RECQL P46063 1/20 0.37
BLM P54132 1/20 0.37
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6676848 0.91 TP53 (0.41) NPC1TP53MAPTTSHRNFKB1
SCHEMBL6675973 0.85 NPC1 (0.40) NPC1TP53MAPTTSHRNFKB1
SCHEMBL7042750 0.83 TP53 (0.43) NPC1TP53MAPTTSHRNFKB1
SCHEMBL6677619 0.83 GAA (0.38) NPC1TP53MAPTTSHRNFKB1
SCHEMBL7039203 0.75 GAA (0.44) POLB
SCHEMBL6673930 0.69 MTTP (0.51) SMN1; SMN2KDM4E
SCHEMBL22129205 0.68 POLB (0.66) NPC1TP53MAPTTSHRNFKB1
SCHEMBL22291931 0.63 NPC1 (0.68) NPC1TP53MAPTNFKB1RAB9A
SCHEMBL5951594 0.62 ACHE (0.47) BACE1ESR1SCN9APARP1
SCHEMBL2367672 0.62 BACE1 (0.58) NPC1RAB9ABACE1POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465613-A2 COMBINATION OF MTP INHIBITORS OR APOB SECRETION INHIBITORS WITH FIBRATES FOR USE AS DRUGS Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2004-10-13 EP disclosed
WO-2003057205-A2 COMBINATION OF MTP INHIBITORS OR APOB SECRETION INHIBITORS WITH FIBRATES FOR USE AS DRUGS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-07-17 WO disclosed
WO-2003004020-A1 HETEROARYL CARBOXYLIC ACID AMIDES, THE PRODUCTION THEREOF AND THE USE OF THE SAME AS INHIBITORS OF THE MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2003-01-16 WO disclosed