SCHEMBL6676182

SCHEMBL6676182

CC/N=C(/NC(=O)OC(C)(C)C)Nc1ccc(CCN)cc1F

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.39
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
NR1H4 Q96RI1 2/20 0.36
KCNQ4 P56696 4/20 0.36
KCNQ5 Q9NR82 4/20 0.36
KCNQ3 O43525 1/20 0.34
KCNQ2 O43526 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ATM Q13315 1/20 0.34
MAPK14 Q16539 1/20 0.33
POLB P06746 1/20 0.33
CTDSP1 Q9GZU7 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KIF11 P52732 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6675309 0.99 CYP17A1 (0.38) CYP17A1CA1CA2NR1H4KCNQ4
Hydrochloric Acid SCHEMBL7242318 0.99 CYP17A1 (0.38) CYP17A1CA1CA2NR1H4KCNQ4
SCHEMBL7248116 0.90 CA1 (0.43) CYP17A1CA1CA2MEN1KMT2A
SCHEMBL6674728 0.79 MEN1 (0.36) CYP17A1MEN1KMT2AATMMAPK14
Hydrochloric Acid SCHEMBL7242320 0.78 MEN1 (0.36) CYP17A1MEN1KMT2AATMMAPK14
SCHEMBL6676258 0.78 CA1 (0.43) CA1CA2NR1H4MEN1KMT2A
SCHEMBL7247586 0.77 CA1 (0.43) CA1CA2MEN1KMT2A
SCHEMBL6681996 0.76 MAPT (0.46) CA1CA2MEN1KMT2AATM
SCHEMBL29468015 0.75 CYP17A1 (0.49) CYP17A1CA1CA2KCNQ4KCNQ5
SCHEMBL16245955 0.74 CYP17A1 (0.48) CYP17A1KCNQ4KCNQ5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP claimed