SCHEMBL6676258

SCHEMBL6676258

CC/N=C(/NC(=O)OC(C)(C)C)Nc1ccc(CCNC(=O)OC(C)(C)C)cc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.43
CA2 P00918 4/20 0.43
PTGER4 P35408 1/20 0.41
NAMPT P43490 1/20 0.41
ALDH1A1 P00352 2/20 0.40
TP53 P04637 2/20 0.39
TSHR P16473 2/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CNR1 P21554 1/20 0.37
NQO2 P16083 1/20 0.37
AKT1 P31749 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7248116 0.89 CA1 (0.43) CA1CA2PTGER4NAMPTKMT2A
SCHEMBL7247586 0.89 CA1 (0.43) CA1CA2PTGER4NAMPTALDH1A1
SCHEMBL6681996 0.88 MAPT (0.46) CA1CA2NAMPTALDH1A1KMT2A
SCHEMBL6676112 0.84 NAMPT (0.54) CA1CA2PTGER4NAMPTKMT2A
SCHEMBL6676262 0.82 PTGER4 (0.41) CA1CA2PTGER4NAMPTALDH1A1
SCHEMBL6688945 0.82 CYP3A4 (0.46) CA1CA2NAMPTNQO2AKT1
SCHEMBL6676121 0.80 CA1 (0.46) CA1CA2PTGER4NAMPTALDH1A1
SCHEMBL6675303 0.80 NQO2 (0.40) ALDH1A1TP53TSHRKMT2AMAPT
SCHEMBL27494819 0.79 NAMPT (0.44) CA1CA2PTGER4NAMPTALDH1A1
SCHEMBL7247902 0.79 NQO2 (0.46) CA1CA2NAMPTALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed