SCHEMBL6676237

SCHEMBL6676237

CN(Cc1ccccc1)c1ccc(N(S)C(N)=O)cc1CN(C(=O)O)C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
STAT5B P51692 1/20 0.35
AKT1 P31749 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
HTR2C P28335 1/20 0.34
SLC6A4 P31645 1/20 0.34
CTSL P07711 2/20 0.33
CTSB P07858 2/20 0.33
CTSS P25774 2/20 0.33
TSHR P16473 1/20 0.33
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
SLC16A3 O15427 1/20 0.32
SLC16A1 P53985 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6679814 0.84 GRM2 (0.33)
SCHEMBL7239503 0.83 GRM2 (0.34)
SCHEMBL6676778 0.80 RXRA (0.35) NR1H2NR1H3
SCHEMBL6677564 0.80 CA12 (0.35) AKT1HDAC3HDAC1HDAC2NCOR2
SCHEMBL6677405 0.80 ACHE (0.39) KEAP1NFE2L2STAT5BAKT1HDAC3
SCHEMBL6676234 0.79 ALDH1A1 (0.39) AKT1HDAC3HDAC1HDAC2NCOR2
SCHEMBL6678485 0.78 GRM2 (0.35)
SCHEMBL6675700 0.78 GRM2 (0.35) HDAC3HDAC1HDAC2NCOR2
SCHEMBL6682109 0.78 STAT5B (0.36) KEAP1NFE2L2STAT5BAKT1HDAC3
SCHEMBL6678438 0.77 GRM2 (0.35) SLC16A3SLC16A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed