SCHEMBL6676262

SCHEMBL6676262

CCNC(=NC(=O)OC(C)(C)C)Nc1ccc(CCNC(=O)OC(C)(C)C)cc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.41
NAMPT P43490 1/20 0.40
ALDH1A1 P00352 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
TP53 P04637 2/20 0.39
TSHR P16473 2/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CNR1 P21554 1/20 0.36
NQO2 P16083 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
HPGD P15428 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
POLB P06746 1/20 0.35
PTPRB P23467 1/20 0.35
GLA P06280 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7248121 0.89 MEN1 (0.41) PTGER4NAMPTALDH1A1CA1CA2
SCHEMBL6675282 0.89 NAMPT (0.40) PTGER4NAMPTALDH1A1CA1CA2
SCHEMBL6681999 0.88 MAPT (0.45) NAMPTALDH1A1CA1CA2KMT2A
SCHEMBL6676115 0.84 NAMPT (0.53) PTGER4NAMPTCA1CA2KMT2A
SCHEMBL6676258 0.82 CA1 (0.43) PTGER4NAMPTALDH1A1CA1CA2
SCHEMBL6675304 0.80 MTNR1A (0.41) MAPTNQO2
SCHEMBL6676121 0.79 CA1 (0.46) PTGER4NAMPTALDH1A1CA1CA2
SCHEMBL27494819 0.78 NAMPT (0.44) PTGER4NAMPTALDH1A1CA1CA2
SCHEMBL6674728 0.77 MEN1 (0.36) KMT2AMEN1TDP1POLB
Hydrochloric Acid SCHEMBL7242320 0.76 MEN1 (0.36) KMT2AMEN1TDP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed