SCHEMBL6676527

SCHEMBL6676527

C#CCN=C(N)Nc1cccc([N+](C)(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HPGD P15428 1/20 0.32
ALDH1A1 P00352 1/20 0.32
PARP14 Q460N5 1/20 0.32
CHIT1 Q13231 3/20 0.31
TDP1 Q9NUW8 1/20 0.31
SIGMAR1 Q99720 6/20 0.31
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
HTR3A P46098 1/20 0.31
HTR3D Q70Z44 1/20 0.31
HTR3C Q8WXA8 1/20 0.31
AURKA O14965 1/20 0.31
RPS6KB1 P23443 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7243106 0.76 SIGMAR1 (0.39) NOS3NOS1NOS2SIGMAR1AURKA
SCHEMBL6676936 0.68 SIGMAR1 (0.45) NOS3NOS1NOS2ALDH1A1SIGMAR1
Hydrochloric Acid SCHEMBL6682202 0.67 SIGMAR1 (0.46) NOS3NOS1NOS2ALDH1A1SIGMAR1
SCHEMBL15171105 0.63 PTGES (0.40) AURKARPS6KB1
SCHEMBL16709846 0.62 HDAC3 (0.43) CA1CA2AURKARPS6KB1
SCHEMBL6678030 0.62 SIGMAR1 (0.44) NOS3NOS1NOS2SIGMAR1GRIN2D
SCHEMBL6676657 0.62 CYP3A4 (0.47) CA1CA2NOS3NOS1NOS2
SCHEMBL6679168 0.61 ADRA2A (0.43) NOS3NOS1NOS2SIGMAR1GRIN2D
SCHEMBL16709841 0.61 HDAC1 (0.42) CA1CA2AURKARPS6KB1
SCHEMBL23455338 0.60 NPC1 (0.48) CA2MEN1KMT2AALDH1A1CHIT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed