SCHEMBL6676770

SCHEMBL6676770

CC(Cc1ccccc1Sc1cccc(OC(=O)c2ccccc2)c1)NC(=O)C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.45
ESR1 P03372 1/20 0.45
CYP2D6 P10635 3/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 2/20 0.39
GPR139 Q6DWJ6 1/20 0.38
GFER P55789 1/20 0.38
TRPV1 Q8NER1 2/20 0.37
TMPRSS15 P98073 1/20 0.37
KMT2A Q03164 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
USP2 O75604 2/20 0.36
CYP3A4 P08684 2/20 0.36
NR1I2 O75469 1/20 0.36
ADRB1 P08588 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6677350 0.89 CYP2D6 (0.45) KCNH2ESR1CYP2D6CYP2C9CYP2C19
SCHEMBL6676499 0.73 ESR1 (0.44) KCNH2ESR1TRPV1SMN1; SMN2PTGDR2
SCHEMBL6676768 0.72 ADRB1 (0.43) KCNH2ESR1CYP2C9SMN1; SMN2ADRB1
SCHEMBL6676771 0.72 ADRB1 (0.43) KCNH2ESR1CYP2C9SMN1; SMN2ADRB1
SCHEMBL6541155 0.71 MTNR1A (0.48) KCNH2ESR1KMT2A
SCHEMBL6676699 0.71 MTNR1A (0.48) KCNH2ESR1KMT2A
SCHEMBL6804630 0.70 ACACB (0.48) KCNH2ESR1CYP2D6CYP2C9KMT2A
SCHEMBL9459072 0.67 ESR1 (0.60) KCNH2ESR1KMT2A
SCHEMBL6677355 0.67 ACACB (0.45) KCNH2ESR1CYP2C9SMN1; SMN2ADRB1
SCHEMBL6677349 0.67 ACACB (0.45) KCNH2ESR1CYP2C9SMN1; SMN2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004045610-A1 AMINOALCOHOL DERIVATIVES AND THEIR USE AS BETA-3 ADRENERGIC RECEPTOR AGONISTS FUJISAWA PHARMACEUTICAL CO., LTD (JP) 2004-06-03 WO disclosed