SCHEMBL6677929

SCHEMBL6677929

CN1CC(Cl)c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.40
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
GPR3 P46089 1/20 0.37
NOTUM Q6P988 1/20 0.37
ACHE P22303 2/20 0.36
HTR2A P28223 3/20 0.36
LMNA P02545 2/20 0.36
ADRA2A P08913 2/20 0.36
ADRA2B P18089 2/20 0.36
ADRA2C P18825 2/20 0.36
SLC6A2 P23975 2/20 0.36
HTR2C P28335 2/20 0.36
SLC6A4 P31645 2/20 0.36
ADRA1A P35348 2/20 0.36
HRH1 P35367 2/20 0.36
HTR2B P41595 2/20 0.36
KCNH2 Q12809 2/20 0.36
MEN1 O00255 2/20 0.36
TP53 P04637 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18681421 0.77 NOTUM (0.55) PAX8MTNR1AMTNR1BGPR3NOTUM
SCHEMBL2625781 0.77 NOTUM (0.55) PAX8MTNR1AMTNR1BGPR3NOTUM
SCHEMBL22240446 0.77 NOTUM (0.55) PAX8MTNR1AMTNR1BGPR3NOTUM
SCHEMBL13372442 0.77 NOTUM (0.55) PAX8MTNR1AMTNR1BGPR3NOTUM
SCHEMBL30509271 0.75 NOTUM (0.41) PAX8MTNR1AMTNR1BGPR3NOTUM
SCHEMBL3702120 0.75 MTNR1A (0.38) PAX8MTNR1AMTNR1BGPR3NOTUM
SCHEMBL27903243 0.75 NOTUM (0.41) PAX8MTNR1AMTNR1BGPR3NOTUM
SCHEMBL21957933 0.75 HTR2A (0.39) PAX8MTNR1AMTNR1BGPR3NOTUM
SCHEMBL19696044 0.73 GPR3 (0.40) PAX8MTNR1AMTNR1BGPR3NOTUM
SCHEMBL29196012 0.73 HTR2A (0.45) PAX8MTNR1AMTNR1BGPR3NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037865-A4 SYNTHESIS OF CC-1065/DUOCARMYCIN ANALOGS SCRIPPS RESEARCH INST (US) 2004-03-31 EP disclosed
US-20020082424-A1 Synthesis of CC-1065/duocarmycin analogs THE SCRIPPS RESEARCH INSTITUTE 2002-06-27 US disclosed
US-6310209-B1 INTERMEDIATES INVOLVED IN THE 5-EXO-TRIG RADICAL CYCLIZATION OF AN ARYL HALIDE ONTO A TETHERED VINYL CHLORIDE FORMING THE DIHYDROINDOLE C-RING WITH CHLORINE INSTALLED AS A SUITABLE LEAVING GROUP FOR SUBSEQUENT CYCLOPROPANE SPIROCYCLIZATION. THE SCRIPPS RESEARCH INSTITUTE 2001-10-30 US disclosed
EP-1037865-A1 SYNTHESIS OF CC-1065/DUOCARMYCIN ANALOGS The Scripps Research Institute (US) 2000-09-27 EP disclosed
WO-1999029642-A1 SYNTHESIS OF CC-1065/DUOCARMYCIN ANALOGS THE SCRIPPS RESEARCH INSTITUTE (US) 1999-06-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020082424-A1 Synthesis of CC-1065/duocarmycin analogs CBR3, C2CD5, SIRT5 PAX8 4461/4885MTNR1A 2118/4885MTNR1B 1801/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.