SCHEMBL6678243

SCHEMBL6678243

COc1ccc(CN2C(=O)c3ccccc3C2=O)cc1[N+](=O)[O-]

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.58
ALDH1A1 P00352 6/20 0.55
LMNA P02545 2/20 0.54
PKM P14618 1/20 0.54
AGTR1 P30556 1/20 0.54
HTT P42858 3/20 0.50
KMT2A Q03164 2/20 0.50
RXFP1 Q9HBX9 2/20 0.50
MEN1 O00255 1/20 0.50
CASP3 P42574 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49
GPR55 Q9Y2T6 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2034683 0.90 RAB9A (0.52) RAB9AALDH1A1LMNAAGTR1HTT
SCHEMBL7073273 0.84 KMT2A (0.51) RAB9AALDH1A1PKMHTTKMT2A
SCHEMBL10924990 0.83 HPGD (0.50) ALDH1A1LMNAPKMAGTR1HTT
SCHEMBL4854039 0.82 NR1H3 (0.62) ALDH1A1LMNAHTTKMT2ARXFP1
SCHEMBL12635556 0.81 ALDH1A1 (0.54) ALDH1A1LMNAPKMHTTKMT2A
SCHEMBL3803546 0.80 HTT (0.53) ALDH1A1HTT
SCHEMBL6679384 0.80 CA12 (0.51) ALDH1A1PKMHTTKMT2AMEN1
SCHEMBL1835526 0.80 HTT (0.50) RAB9AALDH1A1LMNAPKMAGTR1
SCHEMBL101837 0.79 HDAC4 (0.52) RAB9AALDH1A1PKMHTTKMT2A
SCHEMBL7945209 0.79 CASP3 (0.55) LMNAHTTKMT2ARXFP1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed