SCHEMBL6678337

SCHEMBL6678337

FC(F)(F)c1ccccc1-c1nnc(-c2cccc(SCc3ccccc3-c3ccccc3)c2)s1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.38
PPARA Q07869 2/20 0.38
HSD11B1 P28845 2/20 0.38
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
SCN9A Q15858 2/20 0.36
QPCTL Q9NXS2 1/20 0.35
CDK2 P24941 1/20 0.34
AKT1 P31749 1/20 0.34
TACR1 P25103 2/20 0.33
FFAR1 O14842 1/20 0.33
PDCD1 Q15116 2/20 0.33
CD274 Q9NZQ7 2/20 0.33
S1PR1 P21453 1/20 0.33
CTSA P10619 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
HSD17B1 P14061 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6156893 0.86 KMT2A (0.40) PPARGPPARAHSD11B1CDK2AKT1
SCHEMBL6678334 0.74 HTR7 (0.37) PPARGPPARAHSD11B1CA12CA1
SCHEMBL1107921 0.68 SCN9A (0.45) HSD11B1SCN9AHSD17B1
SCHEMBL4955280 0.68 DPP4 (0.44) HSD11B1CA12CA1CA2CA9
SCHEMBL6153697 0.68 CA12 (0.41) HSD11B1CA12CA1CA2CA9
SCHEMBL1107918 0.65 SCN9A (0.42) HSD11B1SCN9A
SCHEMBL2442712 0.64 HSD11B1 (0.54) HSD11B1
SCHEMBL1107958 0.64 SCN9A (0.43) HSD11B1SCN9A
SCHEMBL9654593 0.63 HSD11B1 (0.49) HSD11B1
SCHEMBL8051369 0.63 HSD11B1 (0.49) HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1446110-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES Structural Bioinformatics Inc. (US) 2004-08-18 EP disclosed
WO-2003032916-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES STRUCTURAL BIOINFORMATICS INC. (US) 2003-04-24 WO disclosed