SCHEMBL6679077

SCHEMBL6679077

COc1ccc(N(S)C(N)=O)cc1CN(C)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
ALDH1A1 P00352 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
POLB P06746 1/20 0.37
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
PKM P14618 1/20 0.35
ALOX15 P16050 1/20 0.35
GAA P10253 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTR2C P28335 2/20 0.34
SLC6A4 P31645 2/20 0.34
NPC1 O15118 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HTR2A P28223 1/20 0.33
CACNA1G O43497 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6679037 0.82 ALDH1A1 (0.54) MEN1KMT2AALDH1A1POLBBCHE
SCHEMBL7247260 0.81 KDM4E (0.40) MTNR1AMTNR1BALDH1A1POLBGAA
SCHEMBL7246130 0.80 MEN1 (0.42) MTNR1AMTNR1BMEN1KMT2AALDH1A1
SCHEMBL7239503 0.78 GRM2 (0.34)
SCHEMBL6681940 0.78 PKM (0.35) MTNR1AMTNR1BMEN1KMT2AALDH1A1
SCHEMBL6678485 0.77 GRM2 (0.35)
SCHEMBL6675700 0.77 GRM2 (0.35) NPC1KDM4E
SCHEMBL6678438 0.76 GRM2 (0.35)
SCHEMBL6681810 0.76 GRM2 (0.39) MTNR1AMTNR1BALDH1A1HTR2CSLC6A4
SCHEMBL6679073 0.76 ALDH1A1 (0.49) MEN1KMT2AALDH1A1GAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed