SCHEMBL6679588

SCHEMBL6679588

COc1cc(N)ccc1CCNC(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.48
IDO1 P14902 4/20 0.47
DRD2 P14416 5/20 0.44
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7246127 0.90 NQO2 (0.48) NQO2IDO1DRD2MTNR1AMTNR1B
SCHEMBL2948649 0.87 GAA (0.50) GAAMAPTTSHRMAPK1HTT
SCHEMBL7771175 0.83 NQO2 (0.46) NQO2IDO1DRD2
SCHEMBL6675032 0.83 NQO2 (0.49) NQO2MAPTHTTIDO1ALDH1A1
SCHEMBL6676049 0.83 IDO1 (0.55) NQO2GAAMAPTTSHRHTT
SCHEMBL20968300 0.83 NQO2 (0.51) NQO2HTTIDO1ALDH1A1
SCHEMBL28350815 0.82 MAPT (0.49) NQO2GAAMAPTHTTIDO1
SCHEMBL8419482 0.81 MTNR1A (0.67) NQO2HTTIDO1DRD2MTNR1A
SCHEMBL7244826 0.81 ALDH1A1 (0.54) NQO2GAAIDO1DRD2ALDH1A1
SCHEMBL7449161 0.81 CA12 (0.50) GAAIDO1DRD2MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
CN-1075808-C Aniline derivatives having nitric oxide synthase inhibitory activity CHUGAI PHARMACEUTICAL CO LTD (JP) 2001-12-05 CN disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed