SCHEMBL6680003

SCHEMBL6680003

COc1ccc(NS(=O)(=O)c2cc(F)c(F)cc2F)cc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 6/20 0.58
SMN1; SMN2 Q16637 6/20 0.58
ALDH1A1 P00352 3/20 0.58
HPGD P15428 2/20 0.58
GAA P10253 3/20 0.53
MAPK1 P28482 2/20 0.53
SGK1 O00141 1/20 0.52
CA1 P00915 1/20 0.51
CA2 P00918 1/20 0.51
UBE2N P61088 1/20 0.51
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
ALOX12 P18054 1/20 0.50
PLAU P00749 1/20 0.50
PGR P06401 1/20 0.50
TP53 P04637 1/20 0.49
HTT P42858 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6675225 0.85 LMNA (0.56) LMNASMN1; SMN2ALDH1A1HPGDGAA
SCHEMBL7536270 0.82 LMNA (0.56) LMNASMN1; SMN2ALDH1A1HPGDGAA
SCHEMBL6680012 0.81 LMNA (0.52) LMNASMN1; SMN2ALDH1A1HPGDGAA
SCHEMBL6676773 0.81 LMNA (0.52) LMNASMN1; SMN2ALDH1A1HPGDGAA
SCHEMBL6675270 0.81 LMNA (0.52) LMNASMN1; SMN2ALDH1A1HPGDGAA
SCHEMBL6679367 0.80 ALDH1A1 (0.57) LMNASMN1; SMN2ALDH1A1HPGDGAA
SCHEMBL6674329 0.79 ALDH1A1 (0.58) LMNASMN1; SMN2ALDH1A1HPGDGAA
SCHEMBL97159 0.79 SGK1 (0.44) LMNASMN1; SMN2ALDH1A1HPGDGAA
SCHEMBL7541078 0.79 SMN1; SMN2 (0.51) LMNASMN1; SMN2ALDH1A1HPGDGAA
SCHEMBL23832758 0.78 ALDH1A1 (0.53) LMNASMN1; SMN2ALDH1A1HPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020013496-A1 Benzene compounds as antiproliferative and cholesterol lowering agents AMGEN INC. 2002-01-31 US claimed
EP-1005453-B1 SUBSTITUTED BENZENE COMPOUNDS AS ANTIPROLIFERATIVE LOWERING AGENTS TULARIK INC (US) 2004-10-27 EP disclosed
US-6388131-B2 Benzenesulfonamide compounds, which encompasses the compound batabulin (2-Fluoro-1-methoxy-4-pentafluorophenylsulfonamidobenzene) TULARIK, INC. 2002-05-14 US disclosed
US-20020013496-A1 Benzene compounds as antiproliferative and cholesterol lowering agents AMGEN INC. 2002-01-31 US disclosed
US-6284923-B1 BENZENESULFONIMIDES FOR TREATMENT OF CANCER AND ANTICHOLESTEROL AGENTS TULARIK INC 2001-09-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020013496-A1 Benzene compounds as antiproliferative and cholesterol lowering agents CYP46A1, TGFB1, NR1H2 LMNA 2006/4885SMN1; SMN2 4446/4885ALDH1A1 1173/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.