SCHEMBL6680339

SCHEMBL6680339

COc1ccc(C(=O)Nc2cn(-c3ccccc3)nc2-c2cccs2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.66
MAPT P10636 9/20 0.62
MEN1 O00255 6/20 0.62
KMT2A Q03164 6/20 0.62
TSHR P16473 2/20 0.62
KDM4E B2RXH2 7/20 0.57
LMNA P02545 5/20 0.57
ALDH1A1 P00352 4/20 0.53
HPGD P15428 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
HDAC3 O15379 1/20 0.53
HDAC4 P56524 1/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53
HDAC2 Q92769 1/20 0.53
HDAC10 Q969S8 1/20 0.53
HDAC11 Q96DB2 1/20 0.53
HDAC8 Q9BY41 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6678084 0.89 MAPT (0.72) ADORA3MAPTMEN1KMT2ATSHR
SCHEMBL6677039 0.89 MEN1 (0.59) ADORA3MAPTMEN1KMT2ATSHR
SCHEMBL6684407 0.88 KDM4E (0.70) ADORA3MAPTMEN1KMT2ATSHR
SCHEMBL6676970 0.88 MAPT (0.66) ADORA3MAPTMEN1KMT2ATSHR
SCHEMBL6681714 0.86 ADORA3 (0.61) ADORA3MAPTMEN1KMT2AKDM4E
SCHEMBL6683017 0.85 MAPT (0.68) ADORA3MAPTMEN1KMT2ATSHR
SCHEMBL6679138 0.85 MAPT (0.64) ADORA3MAPTMEN1KMT2ATSHR
SCHEMBL6678678 0.84 ADORA3 (0.60) ADORA3MAPTMEN1KMT2AKDM4E
SCHEMBL6683268 0.81 MAPT (0.62) ADORA3MAPTMEN1KMT2ATSHR
SCHEMBL6686801 0.81 MEN1 (0.71) ADORA3MAPTMEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004043951-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF PEROXISOME PROLIFERATOR ACTIVATED RECEPTORS CAREX S.A. (FR) 2004-05-27 WO claimed
WO-2004043951-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF PEROXISOME PROLIFERATOR ACTIVATED RECEPTORS CAREX S.A. (FR) 2004-05-27 WO disclosed