SCHEMBL6681975

SCHEMBL6681975

CC(C)(C)OC(=O)NN(Cc1cccc(NC(=N)N[N+](=O)[O-])c1)C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.44
MMP1 P03956 2/20 0.41
MMP2 P08253 2/20 0.41
MMP9 P14780 2/20 0.41
MMP8 P22894 2/20 0.41
MMP13 P45452 2/20 0.41
BACE1 P56817 5/20 0.40
AURKA O14965 1/20 0.36
RPS6KB1 P23443 1/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6681977 0.82 AKT1 (0.43) AKT1MMP1MMP2MMP9MMP8
SCHEMBL6679736 0.82 GLS (0.46) MMP1MMP2MMP9MMP8MMP13
SCHEMBL6681292 0.80 AKT1 (0.49) AKT1MMP1MMP2MMP9MMP8
SCHEMBL6681909 0.79 AKT1 (0.51) AKT1MMP1MMP2MMP9MMP8
SCHEMBL6679466 0.77 KDM1A (0.43)
Acetic Acid SCHEMBL6681849 0.75 KDM1A (0.43) BACE1
SCHEMBL6690431 0.75 BACE1 (0.41) AKT1BACE1AURKARPS6KB1
SCHEMBL6676802 0.74 AKT1 (0.55) AKT1BACE1CTSLCTSBCTSS
SCHEMBL6689701 0.74 RXFP1 (0.42) MMP1MMP2MMP9MMP8MMP13
SCHEMBL1402743 0.74 AKT1 (0.57) AKT1CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0798292-B1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY CHUGAI SEIYAKUKABUSHIKI KAISHA (JP) 2004-11-03 EP disclosed
US-6534546-B1 Guanidine- or isothioureido-N-derived anilines; brain, nervous system, and neurodegenerative disorders CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2003-03-18 US disclosed
EP-0798292-A1 ANILINE DERIVATIVES HAVING NITROGEN MONOXIDE SYNTHASE INHIBITORY ACTIVITY Chugai Seiyaku Kabushiki Kaisha (JP) 1997-10-01 EP disclosed