SCHEMBL6683071

SCHEMBL6683071

Nc1ccc(Br)c(Cl)c1-c1nnc(-c2ccc3nonc3c2)s1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.35
MAPT P10636 3/20 0.35
ALDH1A1 P00352 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
SNCA P37840 2/20 0.33
MGAM O43451 1/20 0.32
GAA P10253 1/20 0.32
SI P14410 1/20 0.32
MGAM2 Q2M2H8 1/20 0.32
NOTUM Q6P988 1/20 0.32
QPCT Q16769 1/20 0.32
QPCTL Q9NXS2 1/20 0.32
MAPK1 P28482 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
FABP3 P05413 1/20 0.30
FABP4 P15090 1/20 0.30
FABP5 Q01469 1/20 0.30
APP P05067 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6154986 0.71 GUSB (0.47) KDM4EALDH1A1GAAMEN1KMT2A
SCHEMBL6154609 0.63 GUSB (0.59) KDM4EMAPTALDH1A1L3MBTL1GAA
SCHEMBL3078778 0.62 ENPP2 (0.58) KDM4EALDH1A1MAPK1FABP3FABP4
SCHEMBL16029956 0.60 MAPT (0.38) KDM4EMAPTALDH1A1L3MBTL1GAA
SCHEMBL28897577 0.60 ENPP2 (0.47) ALDH1A1GAAMAPK1MEN1KMT2A
SCHEMBL26092700 0.59 TDO2 (0.40) FABP3FABP4FABP5APP
SCHEMBL30296284 0.58 TDO2 (0.40) KDM4EMAPTALDH1A1FABP3FABP4
SCHEMBL980630 0.56 MAP4K4 (0.50) KDM4EMAPTALDH1A1GAAMEN1
SCHEMBL3191645 0.55 ENPP2 (0.54) KDM4EMAPTALDH1A1GAAMEN1
SCHEMBL298552 0.55 ENPP2 (0.54) ALDH1A1MAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1446110-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES Structural Bioinformatics Inc. (US) 2004-08-18 EP disclosed
WO-2003032916-A2 ORGANOSULFUR INHIBITORS OF TYROSINE PHOSPHATASES STRUCTURAL BIOINFORMATICS INC. (US) 2003-04-24 WO disclosed