SCHEMBL6683586

SCHEMBL6683586

C1=C(CNCCc2ccccc2)c2ccccc2C1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.53
MAPT P10636 1/20 0.53
HTR6 P50406 1/20 0.46
MPO P05164 1/20 0.45
SIGMAR1 Q99720 7/20 0.44
HTR2A P28223 1/20 0.44
HRH1 P35367 1/20 0.44
GRIN2B Q13224 1/20 0.42
BCHE P06276 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23023190 0.87 GAA (0.53) GAAMAPTHTR6MPOSIGMAR1
SCHEMBL28220073 0.81 HTR6 (0.53) GAAMAPTHTR6SIGMAR1HTR2A
SCHEMBL6666864 0.80 HTR6 (0.45) MAPTHTR6HTR2AHRH1
SCHEMBL6664305 0.76 HTR6 (0.42) HTR6
SCHEMBL6683869 0.76 HTR6 (0.47) GAAHTR6HTR2AALDH1A1
SCHEMBL10849661 0.76 GAA (0.47) GAAMAPTMPOSIGMAR1BCHE
SCHEMBL6130448 0.75 HTR6 (0.74) GAAMAPTHTR6SIGMAR1MEN1
SCHEMBL31121639 0.74 HTR6 (0.56) HTR6SIGMAR1BCHECA12CA9
SCHEMBL2338975 0.74 HTR6 (0.56) HTR6SIGMAR1BCHECA12CA9
SCHEMBL1604010 0.73 HTR6 (0.45) HTR6SIGMAR1HTR2AHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1359916-A4 IMIDAZOLYL DERIVATIVES AS CORTICOTROPIN RELEASING FACTOR INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2004-04-07 EP disclosed
EP-1359916-A1 IMIDAZOLYL DERIVATIVES AS CORTICOTROPIN RELEASING FACTOR INHIBITORS Bristol-Myers Squibb Company (US) 2003-11-12 EP disclosed
WO-2002058704-A1 IMIDAZOLYL DERIVATIVES AS CORTICOTROPIN RELEASING FACTOR INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2002-08-01 WO disclosed