SCHEMBL6683695

SCHEMBL6683695

O=C(O)C1C(O)CN1C(=O)OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 5/20 0.55
SMN1; SMN2 Q16637 2/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
PSEN1 P49768 1/20 0.49
PSEN2 P49810 1/20 0.49
APH1B Q8WW43 1/20 0.49
NCSTN Q92542 1/20 0.49
APH1A Q96BI3 1/20 0.49
PSENEN Q9NZ42 1/20 0.49
HTR2C P28335 1/20 0.48
CYP2C19 P33261 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
POLB P06746 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
PDK1 Q15118 1/20 0.45
PDK2 Q15119 1/20 0.45
PDK3 Q15120 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9175852 0.92 AGTR2 (0.53) AGTR2SMN1; SMN2NPC1RAB9APSEN1
SCHEMBL9175859 0.92 AGTR2 (0.53) AGTR2SMN1; SMN2NPC1RAB9APSEN1
SCHEMBL6285084 0.90 AGTR2 (0.52) AGTR2SMN1; SMN2NPC1RAB9APSEN1
SCHEMBL6343357 0.90 AGTR2 (0.52) AGTR2SMN1; SMN2NPC1RAB9APSEN1
SCHEMBL16256994 0.89 AGTR2 (0.51) AGTR2SMN1; SMN2NPC1RAB9APSEN1
SCHEMBL21359881 0.89 AGTR2 (0.51) AGTR2SMN1; SMN2NPC1RAB9APSEN1
SCHEMBL3431539 0.89 AGTR2 (0.51) AGTR2SMN1; SMN2NPC1RAB9APSEN1
SCHEMBL14763059 0.88 AGTR2 (0.50) AGTR2SMN1; SMN2NPC1RAB9APSEN1
SCHEMBL9763260 0.88 AGTR2 (0.50) AGTR2SMN1; SMN2NPC1RAB9APSEN1
SCHEMBL21874593 0.87 SMN1; SMN2 (0.58) AGTR2SMN1; SMN2NPC1RAB9ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004071454-A2 SUBSTITUTED AZETIDINE COMPOUNDS AS INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARMACEUTICALS INC. (US) 2004-08-26 WO disclosed